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3-(6-Methyl-pyridazin-3-yloxy)-piperidine-1-carboxylic acid tert-butylester

3-Methyl-6-(piperidin-3-yloxy)-pyridazine hydrochloride

3-Methyl-6-(piperidin-4-yloxy)-pyridazine hydrochloride

3-Methyl-6-(piperidin-3-ylmethoxy)-pyridazine hydrochloride

3-Methyl-6-(piperidin-4-ylmethoxy)-pyridazine hydrochloride

3-(6-Chloro-pyridazin-3-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

(6-Chloro-pyridazin-3-yl)-pyrrolidin-3-yl-amine hydrochloride

(S)-3-(6-Chloro-pyridazin-3-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-Bromo-pyridine

(6-Chloro-pyridazin-3-yl)-(S)-pyrrolidin-3-yl-amine hydrochloride

2-Chloro-nicotinonitrile

(R)-3-(6-Chloro-pyridazin-3-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

(6-Chloro-pyridazin-3-yl)-(R)-pyrrolidin-3-yl-amine hydrochloride

(6-Chloro-pyridazin-3-yl)-pyrrolidin-2-ylmethyl-amine hydrochloride

1-(6-Chloro-pyridazin-3-yl)-azetidine-3-carboxylic acid

4-(6-Chloro-pyridazin-3-yl)-piperazine-2-carboxylic acid

4-(6-Chloro-pyridazin-3-yl)-3-methyl-piperazine-1-carboxylic acid tert-butyl ester

3-Chloro-6-(2-methyl-piperazin-1-yl)-pyridazine hydrochloride

3-Chloro-6-(3-methyl-piperazin-1-yl)-pyridazine hydrochloride

4-(6-Chloro-pyridazin-3-yl)-piperazine-1,3-dicarboxylic acid 1-tert-butyl ester

1-(6-Chloro-pyridazin-3-yl)-piperazine-2-carboxylic acid hydrochloride

2,4-Dichloro-pyrimidine

4-Chloro-pyridine hydrochloride

2-Bromo-4-methyl-pyridine

[1-(6-Chloro-pyridazin-3-yl)-piperidin-4-yl]-methyl-amine hydrochloride

(6-Chloro-pyridazin-3-yl)-methyl-piperidin-3-yl-amine hydrochloride

3-Chloro-6-(pyrrolidin-2-ylmethoxy)-pyridazine hydrochloride

3-Chloro-6-(piperidin-2-ylmethoxy)-pyridazine hydrochloride

3-Chloro-6-(piperidin-4-ylmethoxy)-pyridazine hydrochloride

[4-(6-Chloro-pyridazin-3-ylamino)-cyclohexyl]-carbamic acid tert-butyl ester

(1r,4r)-N1-(6-chloropyridazin-3-yl)cyclohexane-1,4-diamine hydrochloride

(1r,4r)-4-(6-chloropyridazin-3-ylamino)cyclohexanol

N-(6-Chloro-pyridazin-3-yl)-cyclohexane-1,4-diamine hydrochloride

[2-(6-Chloro-pyridazin-3-ylamino)-cyclohexyl]-carbamic acid tert-butyl ester

N-(6-Chloro-pyridazin-3-yl)-cyclohexane-1,2-diamine hydrochloride

2-(4-chloropiperidin-1-yl)isonicotinonitrile

2-(4-chloropiperidin-1-yl)nicotinonitrile

1-(1-(pyridin-2-yl)ethyl)piperazine hydrochloride

tert-butyl4-(6-(2-acetyl-1H-pyrrol-1-yl)pyridin-2-yl)piperazine-1-carboxylate

1-(1-(pyridin-2-yl)-1H-pyrrol-2-yl)ethanone

2-chloro-5-((4-chloropiperidin-1-yl)methyl)pyridine

2-(2-Bromo-pyridin-3-yloxy)-pyrimidine

Bis-(6-chloro-pyridin-3-ylmethyl)-cyclopropyl-amine

5-methyl-N-(piperidin-4-yl)pyridin-2-mine hydrochloride

1-(1-(pyridin-2-yl)ethyl)piperidin-4-amine hydrochloride

5-methyl-N-(piperidin-3-ylmethyl)pyridin-2-amine hydrochloride

N-(piperidin-3-ylmethyl)pyridin-2-amine hydrochloride

(3-Chloro-5-trifluoromethyl-pyridin-2-yl)-piperidin-4-yl-amine hydrochloride

2-Bromo-3-(pyridin-2-ylmethoxy)-pyridine

2-Bromo-3-(pyridin-3-ylmethoxy)-pyridine

2-Bromo-3-(pyridin-4-ylmethoxy)-pyridine

2-Bromo-3-(thiazol-2-yloxy)-pyridine

2-Bromo-3-(pyridin-2-yloxy)-pyridine

2-(2-Bromo-pyridin-3-yloxy)-pyrazine

2-bromo-6-(2-bromopyridin-3-yloxy)pyridine

2-(2-bromopyridin-3-yloxy)-5-(chloromethyl)pyridine

2-(2-Bromo-pyridin-3-yloxy)-4-chloro-pyrimidine

4-(2-Bromo-pyridin-3-yloxy)-6-chloro-pyrimidine

2-Bromo-3-(5-chloromethyl-thiazol-2-yloxy)-pyridine

3-(2-Bromo-pyridin-3-yloxy)-6-chloro-pyridazine

2-(2-Bromo-pyridin-3-yloxy)-3-chloro-quinoxaline

2-(2-Bromo-pyridin-3-yloxy)-benzothiazole

2-(2-Bromo-pyridin-3-yloxy)-nicotinonitrile

2-(2-Bromo-pyridin-3-yloxy)-isonicotinonitrile

2-Chloro-N-(3 -cyano-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-yl)-acetamide

2-Chloro-N-(3 -cyano-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-yl)-acetamide

2-Chloro-N-(4 -cyano-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-yl)-acetamide

2-Chloro-N-(3 -nitro-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-yl)-acetamide

2-Chloro-N-(3 -nitro-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-yl)-acetamide

2-Bromo-6-(furan-2-ylmethoxy)-pyridine

2-(Furan-2-ylmethoxy)-3-nitro-pyridine

2-(Furan-2-ylmethoxy)-5-nitro-pyridine

5-Chloromethyl-2-(furan-2-ylmethoxy)-pyridine

3 -Chloro-5 -trifluoromethyl-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-ylamine hydrochloride

(3-Chloro-5-trifluoromethyl-pyridin-2-yl)-piperidin-4-ylmethyl-amine hydrochloride

3 -Chloro-5 -trifluoromethyl-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-ylamine hydrochloride

(3-Chloro-5-trifluoromethyl-pyridin-2-yl)-piperidin-3-yl-amine hydrochloride

(3-Chloro-5-trifluoromethyl-pyridin-2-yl)-piperidin-3-ylmethyl-amine hydrochloride

2-Chloro-N-(5-nitro-pyridin-2-yl)-acetamide

2-Chloro-N-(3-nitro-pyridin-2-yl)-acetamide

5 -Nitro-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl

3-Nitro-2-(piperidin-4-yloxy)-pyridine hydrochloride

4-(3-Nitro-pyridin-2-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

3-Nitro-2-(piperidin-3-yloxy)-pyridine hydrochloride

3-(3-Nitro-pyridin-2-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

3-Nitro-2-(piperidin-3-ylmethoxy)-pyridine hydrochloride

3-(3-Nitro-pyridin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

4-(3-Cyano-pyridin-2-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

4-Methyl-2-(piperidin-4-yloxy)-pyridine hydrochloride

4-(4-Methyl-pyridin-2-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

4-Methyl-2-(piperidin-3-yloxy)-pyridine hydrochloride

3-(4-Methyl-pyridin-2-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

4-Methyl-2-(piperidin-3-ylmethoxy)-pyridine hydrochloride

3-(4-Methyl-pyridin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-Chloro-N-(3-cyano-pyridin-2-yl)-acetamide

1-(6-Methoxy-pyridin-3-ylmethyl)-piperidin-3-ylamine dihydrochloride

4-(5-Nitro-pyridin-2-yl)-morpholine

4-(3-Nitro-pyridin-2-yl)-morpholine

1-(6-Methoxy-pyridin-3-ylmethyl)-piperidin-4-ylamine dihydrochloride

1-(6-Ethoxy-pyridin-3-ylmethyl)-piperidin-4-ylamine dihydrochloride

6 -Bromo-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-carboxylic acid

(6 -Bromo-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-yl)-methanol

6 -Bromo-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-ylamine hydrochloride

(6 -Bromo-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-yl)-carbamic acid tert-butyl ester

6 -Bromo-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-ylamine hydrochloride

(6 -Bromo-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-yl)-carbamic acid tert-butyl ester

(6-Bromo-pyridin-2-yl)-piperidin-4-yl-amine hydrochloride

4-(6-Bromo-pyridin-2-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

(6-Bromo-pyridin-2-yl)-piperidin-3-yl-amine hydrochloride

3-(6-Bromo-pyridin-2-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

(6-Bromo-pyridin-2-yl)-piperidin-4-ylmethyl-amine hydrochloride

4-[(6-Bromo-pyridin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

(6-Bromo-pyridin-2-yl)-piperidin-3-ylmethyl-amine hydrochloride

3-[(6-Bromo-pyridin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

2-Bromo-6-(piperidin-4-yloxy)-pyridine hydrochloride

4-(6-Bromo-pyridin-2-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

2-Bromo-6-(piperidin-3-yloxy)-pyridine hydrochloride

3-(6-Bromo-pyridin-2-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

2-Bromo-6-(piperidin-3-ylmethoxy)-pyridine hydrochloride

3-(6-Bromo-pyridin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

(3-Nitro-pyridin-2-yl)-piperidin-4-yl-amine hydrochloride

4-(6-Chloro-pyridin-3-ylmethyl)-piperazine-1-carboxylic acid tert-butyl ester

(5 -Nitro-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-yl)-methanol

4 -Methyl-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-ylamine hydrochloride

1-(5-nitropyridin-2-yl)-piperazine hydrochloride

1-(5-nitropyridin-2-yl)-3-piperidinamine hydrochloride

(3-Nitro-pyridin-2-yl)-piperidin-3-ylmethyl-amine hydrochloride

(1-Pyridin-3-ylmethyl-piperidin-3-yl)-methanol dihydrochloride

1-Pyridin-3-ylmethyl-piperidin-3-ylamine dihydrochloride

3 -Nitro-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-ylamine hydrochloride

1-(3-Nitro-pyridin-2-yl)-piperazine hydrochloride

4-(6-Chloro-pyridin-3-ylmethoxy)-piperidine-1-carboxylic acid tert-butyl ester

3 -Nitro-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-ylamine hydrochloride

3,4,5,6-Tetrahydro-2H-[1,2 ]bipyridinyl-4,3 -dicarboxylic acid 3 -methyl ester hydrochloride

2-[(Piperidin-3-ylmethyl)-amino]-nicotinic acid methyl ester dihydrochloride

4-(3-Nitro-pyridin-2-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

3-(3-Nitro-pyridin-2-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

3-Hydroxymethyl-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4 -carbonitrile

4-(3-Nitro-pyridin-2-yl)-piperazine-1-carboxylic acid tert-butyl ester

4-Hydroxy-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3 -carbonitrile

1-(3-Nitro-pyridin-2-yl)-[1,4]diazepane

1-(4-Methyl-pyridin-2-yl)-piperazine hydrochloride

(3,4,5,6-Tetrahydro-2H-[1,2 ]bipyridinyl-3-yl)-methanol

3-Hydroxy-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3 -carbonitrile

5 -Nitro-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-ylamine hydrochloride

(3 -Nitro-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-yl)-carbamic acid tert-butyl ester

1-Pyridin-3-ylmethyl-piperazine dihydrochloride

3,4,5,6-Tetrahydro-2H-[1,2 ]bipyridinyl-4-carboxylic acid

4-Amino-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4 -carbonitrile hydrochloride

4-Hydroxy-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3 -carboxylic acid methyl ester hydrochloride

2-(Piperidin-3-ylmethoxy)-pyridine hydrochloride

(3-Nitro-pyridin-2-yl)-piperidin-3-yl-amine hydrochloride

2-(Piperidin-4-yloxy)-pyridine hydrochloride

4-(4-Chloro-benzenesulfinylmethyl)-piperidine

3-(4-Chloro-benzenesulfinylmethyl)-piperidine

2-(4-Chloro-benzenesulfinylmethyl)-piperidine

4-(4-Chloro-benzenesulfinyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(4-Chloro-benzenesulfinyl)-piperidine-1-carboxylic acid tert-butyl ester

4-(4-Chloro-benzenesulfinylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(4-Chloro-benzenesulfinylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-(4-Chloro-benzenesulfinylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

(S)-3-(4-Chloro-benzenesulfonyl)-pyrrolidine

(R)-3-(4-Chloro-benzenesulfonyl)-pyrrolidine

3-(4-Chloro-benzenesulfonyl)-pyrrolidine

3-(4-Chloro-benzenesulfonylmethyl)-pyrrolidine

2-(4-Chloro-benzenesulfonylmethyl)-pyrrolidine

(S)-3-(4-Chloro-benzenesulfonyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

(R)-3-(4-Chloro-benzenesulfonyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(4-Chloro-benzenesulfonyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(4-Chloro-benzenesulfonylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-(4-Chloro-benzenesulfonylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

4-(4-Chloro-benzenesulfonyl)-piperidine

3-(4-Chloro-benzenesulfonyl)-piperidine

4-(4-Chloro-benzenesulfonylmethyl)-piperidine

3-(4-Chloro-benzenesulfonylmethyl)-piperidine

2-(4-Chloro-benzenesulfonylmethyl)-piperidine

4-(4-Chloro-benzenesulfonyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(4-Chloro-benzenesulfonyl)-piperidine-1-carboxylic acid tert-butyl ester

4-(4-Chloro-benzenesulfonylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(4-Chloro-benzenesulfonylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-(4-Chloro-benzenesulfonylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

(R)-3-(4-Nitro-phenylsulfanyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(4-Nitro-phenylsulfanyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(4-Nitro-phenylsulfanyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(4-Nitro-phenylsulfanylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-(4-Nitro-phenylsulfanylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

(R)-3-(4-Nitro-phenylsulfanyl)-pyrrolidine

(S)-3-(4-Nitro-phenylsulfanyl)-pyrrolidine

3-(4-Nitro-phenylsulfanyl)-pyrrolidine

3-(4-Nitro-phenylsulfanylmethyl)-pyrrolidine

3-Hydroxymethyl-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3 -carbonitrile

1-(6-Chloro-pyridin-3-ylmethyl)-piperidin-4-ylamine dihydrochloride

2-(4-Nitro-phenylsulfanylmethyl)-pyrrolidine

2-Chloro-5-(piperidin-3-ylmethoxymethyl)-pyridine dihydrochloride

4-(4-Nitro-phenylsulfanyl)-piperidine

3-(4-Nitro-phenylsulfanyl)-piperidine

2-(Piperidin-3-ylamino)-nicotinic acid methyl ester dihydrochloride

4-(4-Nitro-phenylsulfanylmethyl)-piperidine

1-Pyridin-4-ylmethyl-piperazine dihydrochloride

3-(4-Nitro-phenylsulfanylmethyl)-piperidine

3 -Cyano-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-carboxylic acid

2-(4-Nitro-phenylsulfanylmethyl)-piperidine

2-(Piperidin-4-ylamino)-nicotinonitrile hydrochloride

2-(Piperidin-3-ylamino)-nicotinonitrile hydrochloride

4-(4-Nitro-phenylsulfanyl)-piperidine-1-carboxylic acid tert-butyl ester

3-Amino-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3 -carboxylic acid methyl ester dihydrochloride

3-(4-Nitro-phenylsulfanyl)-piperidine-1-carboxylic acid tert-butyl ester

1-Pyridin-2-yl-piperazine hydrochloride

4-(4-Nitro-phenylsulfanylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

1-(6-Chloro-pyridin-3-ylmethyl)-piperidin-3-ylamine dihydrochloride

3-(4-Nitro-phenylsulfanylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-Piperazin-1-yl-nicotinonitrile hydrochloride

3 -Nitro-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-ol

2-(4-Nitro-phenylsulfanylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-Chloro-5-(piperidin-4-yloxymethyl)-pyridine dihydrochloride

(S)-3-(4-Nitro-benzenesulfinyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(3-Cyano-pyridin-2-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

(R)-3-(4-Nitro-benzenesulfinyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3,4,5,6-Tetrahydro-2H-[1,2 ]bipyridinyl-3-ylamine hydrochloride

3,4,5,6-Tetrahydro-2H-[1,2 ]bipyridinyl-4-ol

3-(4-Nitro-benzenesulfinyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

4-[(3-Cyano-pyridin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

2-(4-Nitro-benzenesulfinylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-(Piperidin-3-yloxy)-pyridine hydrochloride

(3-Nitro-pyridin-2-yl)-piperidin-4-ylmethyl-amine hydrochloride

(R)-3-(4-Nitro-benzenesulfinyl)-pyrrolidine

4-(3-Cyano-pyridin-2-yl)-piperazine-1-carboxylic acid tert-butyl ester

(S)-3-(4-Nitro-benzenesulfinyl)-pyrrolidine

3-(4-Nitro-benzenesulfinyl)-pyrrolidine

3-(4-Nitro-benzenesulfinylmethyl)-pyrrolidine

2-(4-Nitro-benzenesulfinylmethyl)-pyrrolidine

4-(4-Nitro-benzenesulfinyl)-piperidine

3-(4-Nitro-benzenesulfinyl)-piperidine

4-(4-Nitro-benzenesulfinylmethyl)-piperidine

5 -Methyl-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-ol

1-Pyridin-3-ylmethyl-piperidin-3-ol dihydrochloride

3 -Nitro-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-carboxylic acid

4-Amino-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3 -carbonitrile hydrochloride

4-(3-Cyano-pyridin-2-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

5 -Methyl-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-ol

(5 -Methyl-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-yl)-methanol

(3 -Cyano-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-yl)-carbamic acid tert-butyl ester

5-Methyl-2-(piperidin-3-yloxy)-pyridine hydrochloride

3 -Nitro-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-ol

5-Methyl-2-(piperidin-3-ylmethoxy)-pyridine hydrochloride

1-(5-Methyl-pyridin-2-yl)-piperazine hydrochloride

5 -Methyl-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-ylamine hydrochloride

5-Methyl-2-(piperidin-4-yloxy)-pyridine hydrochloride

5-Nitro-2-(piperidin-4-yloxy)-pyridine hydrochloride

3-[(3-Cyano-pyridin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

3,4,5,6-Tetrahydro-2H-[1,2 ]bipyridinyl-3-ol

5 -Methyl-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-ylamine hydrochloride

5-Nitro-2-(piperidin-3-ylmethoxy)-pyridine hydrochloride

(3 -Nitro-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-yl)-methanol

3-(5-Nitro-pyridin-2-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

4 -Methyl-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-ol

4-(5-Methyl-pyridin-2-yl)-piperazine-1-carboxylic acid tert-butyl ester

(5 -Methyl-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-yl)-carbamic acid tert-butyl ester

(5 -Methyl-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-yl)-carbamic acid tert-butyl ester

4-(5-Nitro-pyridin-2-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

4 -Methyl-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-ol

3-(5-Nitro-pyridin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

4 -Methyl-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-ylamine hydrochloride

[1-(6-Chloro-pyridin-3-ylmethyl)-piperidin-3-yl]-carbamic acid tert-butyl ester

(4-Methyl-pyridin-2-yl)-piperidin-3-yl-amine hydrochloride

4-(5-Methyl-pyridin-2-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

3-(5-Methyl-pyridin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

[1-(6-Chloro-pyridin-3-ylmethyl)-piperidin-3-yl]-methanol dihydrochloride

4-(4-Methyl-pyridin-2-yl)-piperazine-1-carboxylic acid tert-butyl ester

(4 -Methyl-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-yl)-methanol

(4 -Methyl-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-yl)-carbamic acid tert-butyl ester

3-[(3-Nitro-pyridin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

4-(4-Methyl-pyridin-2-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

(4 -Cyano-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-yl)-carbamic acid tert-butyl ester

(4 -Methyl-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-yl)-carbamic acid tert-butyl ester

4 -Cyano-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-carboxylic acid

5-Nitro-2-(piperidin-3-yloxy)-pyridine hydrochloride

3-Amino-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4 -carbonitrile hydrochloride

(3 -Nitro-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-yl)-carbamic acid tert-butyl ester

4-(4-Cyano-pyridin-2-yl)-piperazine-1-carboxylic acid tert-butyl ester

2-[(Piperidin-4-ylmethyl)-amino]-nicotinic acid methyl ester dihydrochloride

(4 -Cyano-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-yl)-carbamic acid tert-butyl ester

1-(6-Chloro-pyridin-3-ylmethyl)-piperidin-4-ol

3-(4-Methyl-pyridin-2-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

1-(6-Chloro-pyridin-3-ylmethyl)-piperidin-3-ol dihydrochloride

4-[(3-Nitro-pyridin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

(3 -Cyano-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-yl)-carbamic acid tert-butyl ester

1-(6-Chloro-pyridin-3-ylmethyl)-piperazine dihydrochloride

(1-Pyridin-4-ylmethyl-piperidin-3-yl)-methanol

2-[(Piperidin-3-ylmethyl)-amino]-nicotinonitrile hydrochloride

(5-Nitro-pyridin-2-yl)-piperidin-3-yl-amine

3-(6-Chloro-pyridin-3-ylmethoxy)-piperidine-1-carboxylic acid tert-butyl ester

3-Hydroxymethyl-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3 -carboxylic acid methyl ester hydrochloride

4-[(4-Methyl-pyridin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

2-Piperazin-1-yl-pyridin-3-ol hydrochloride

2-[(Piperidin-4-ylmethyl)-amino]-nicotinonitrile hydrochloride

1-Pyridin-2-ylmethyl-piperidin-3-ol

2-Chloro-5-(piperidin-3-yloxymethyl)-pyridine dihydrochloride

3-Amino-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3 -carbonitrile hydrochloride

(1-Pyridin-2-ylmethyl-piperidin-3-yl)-methanol

(5-Nitro-pyridin-2-yl)-piperidin-4-yl-amine

(5-Nitro-pyridin-2-yl)-piperidin-4-ylmethyl-amine

2-(Piperidin-4-yloxymethyl)-pyridine dihydrochloride

4-Hydroxy-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4 -carbonitrile

2-(Piperidin-3-ylmethoxymethyl)-pyridine dihydrochloride

1-Pyridin-2-ylmethyl-piperidin-3-ylamine dihydrochloride

3-(6-Chloro-pyridin-3-ylmethoxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

(4-Methyl-pyridin-2-yl)-piperidin-4-yl-amine hydrochloride

(5-nitro-pyridin-2-yl)-piperidin-3-ylmethyl-amine

2-Piperazin-1-yl-isonicotinonitrile hydrochloride

1-Pyridin-2-ylmethyl-piperazine dihydrochloride

1-Pyridin-3-ylmethyl-piperidin-4-ol dihydrochloride

2-[(Piperidin-4-ylmethyl)-amino]-nicotinic acid methyl ester compoundwith trifluoro-acetic acid

[1-(6-Chloro-pyridin-3-ylmethyl)-piperidin-4-yl]-carbamic acid tert-butyl ester

3-[(4-Methyl-pyridin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

3-(Piperidin-4-yloxymethyl)-pyridine dihydrochloride

2-Piperazin-1-yl-nicotinic acid methyl ester dihydrochloride

(4-Methyl-pyridin-2-yl)-piperidin-4-ylmethyl-amine hydrochloride

5 -Nitro-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-ol

3-(Piperidin-3-ylmethoxymethyl)-pyridine dihydrochloride

1-Pyridin-4-ylmethyl-piperidin-4-ol

3-Hydroxy-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4 -carbonitrile

5 -Nitro-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-carboxylic acid

1-Pyridin-4-ylmethyl-piperidin-3-ol

(4-Methyl-pyridin-2-yl)-piperidin-3-ylmethyl-amine hydrochloride

4-Amino-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3 -carboxylic acid methyl ester dihydrochloride

5 -Nitro-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-ol

3-(4-Nitro-benzenesulfinylmethyl)-piperidine

1-Pyridin-2-ylmethyl-piperidin-4-ol

3-(5-Methyl-pyridin-2-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

2-(4-Nitro-benzenesulfinylmethyl)-piperidine

1-Pyridin-4-ylmethyl-piperidin-3-ylamine dihydrochloride

4-(4-Nitro-benzenesulfinyl)-piperidine-1-carboxylic acid tert-butyl ester

4-(6-Chloro-pyridin-3-ylmethoxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

4-(6-Bromo-pyridin-2-yl)-piperazine-1,3-dicarboxylic acid 1-tert-butylester

3-(4-Nitro-benzenesulfinyl)-piperidine-1-carboxylic acid tert-butyl ester

5-Nitro-2-(piperidin-2-ylmethoxy)-pyridine hydrochloride

4-(4-Nitro-benzenesulfinylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-(3-Nitro-pyridin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(4-Nitro-benzenesulfinylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-Nitro-2-(piperidin-4-ylmethoxy)-pyridine hydrochloride

4-(3-Cyano-pyridin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-(4-Nitro-benzenesulfinylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

(R)-3-(4-Nitro-benzenesulfonyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

4-(Pyridin-2-ylmethoxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

(6 -Bromo-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-yl)-methanol

(S)-3-(4-Nitro-benzenesulfonyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

6 -Bromo-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-2-carboxylic acid

3-(4-Nitro-benzenesulfonyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

6 -Bromo-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-carboxylic acid

3-(4-Nitro-benzenesulfonylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

(1r,4r)-4-((6-chloropyridin-3-yl)methylamino)cyclohexanol

2-(4-Nitro-benzenesulfonylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

(1r,4r)-4-(3-nitropyridin-2-ylamino)cyclohexanol

(1r,4r)-4-(5-nitropyridin-2-ylamino)cyclohexanol

(R)-3-(4-Nitro-benzenesulfonyl)-pyrrolidine

2-{[(6-Chloro-pyridin-3-ylmethyl)-amino]-methyl}-pyrrolidine-1-carboxylic acid tert-butyl ester

S)-3-(4-Nitro-benzenesulfonyl)-pyrrolidine

(S)-3-(6-Chloro-pyridin-3-ylmethoxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(4-Nitro-benzenesulfonyl)-pyrrolidine

(R)-3-(6-Chloro-pyridin-3-ylmethoxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(4-Nitro-benzenesulfonylmethyl)-pyrrolidine

2-Chloro-5-((R)-pyrrolidin-3-yloxymethyl)-pyridine hydrochloride

2-(4-Nitro-benzenesulfonylmethyl)-pyrrolidine

4-(6-Chloro-pyridin-3-ylmethyl)-3-methyl-piperazine-1-carboxylic acid tert-butyl ester

4-(4-Nitro-benzenesulfonyl)-piperidine

1-(6-Chloro-pyridin-3-ylmethyl)-2-methyl-piperazine hydrochloride

4-(6-Chloro-pyridin-3-ylmethyl)-2-methyl-piperazine-1-carboxylic acid tert-butyl ester

3-(4-Nitro-benzenesulfonyl)-piperidine

1-(6-Chloro-pyridin-3-ylmethyl)-3-methyl-piperazine hydrochloride

4-(4-Nitro-benzenesulfonylmethyl)-piperidine

[1-(6-Chloro-pyridin-3-ylmethyl)-piperidin-4-yl]-methyl-carbamic acid tert-butyl ester

2-(6-Chloro-pyridin-3-ylmethoxymethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(4-Nitro-benzenesulfonylmethyl)-piperidine

3-[(6-Chloro-pyridin-3-ylmethyl)-methyl-amino]-piperidine-1-carboxylic acid tert-butyl ester

2-(4-Nitro-benzenesulfonylmethyl)-piperidine

(6-Chloro-pyridin-3-ylmethyl)-methyl-piperidin-3-yl-amine hydrochloride

4-(4-Nitro-benzenesulfonyl)-piperidine-1-carboxylic acid tert-butyl ester

[1-(6-Chloro-pyridin-3-ylmethyl)-piperidin-3-yl]-methyl-carbamic acid tert-butyl ester

3-(4-Nitro-benzenesulfonyl)-piperidine-1-carboxylic acid tert-butyl ester

[1-(6-Chloro-pyridin-3-ylmethyl)-piperidin-3-yl]-methyl-amine hydrochloride

4-(4-Nitro-benzenesulfonylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(4-Cyano-pyridin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butylester

3-(4-Nitro-benzenesulfonylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-[(Pyrrolidin-2-ylmethyl)-amino]-isonicotinonitrile hydrochloride

2-(4-Nitro-benzenesulfonylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-(3-Hydroxy-pyrrolidin-1-yl)-isonicotinonitrile

2-((S)-3-Hydroxy-pyrrolidin-1-yl)-isonicotinonitrile

(R)-3-(4-Bromo-phenylsulfanyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-((R)-3-Hydroxy-pyrrolidin-1-yl)-isonicotinonitrile

(S)-3-(4-Bromo-phenylsulfanyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(4-Bromo-phenylsulfanyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(4-Bromo-phenylsulfanylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-(4-Bromo-phenylsulfanylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(4-Bromo-phenylsulfanyl)-pyrrolidine

3-(4-Bromo-phenylsulfanyl)-pyrrolidine

3-(4-Bromo-phenylsulfanylmethyl)-pyrrolidine

2-(4-Bromo-phenylsulfanylmethyl)-pyrrolidine

4-(4-Bromo-phenylsulfanyl)-piperidine

3-(4-Bromo-phenylsulfanyl)-piperidine

4-(4-Bromo-phenylsulfanylmethyl)-piperidine

3-(4-Bromo-phenylsulfanylmethyl)-piperidine

2-(4-Bromo-phenylsulfanylmethyl)-piperidine

4-(4-Bromo-phenylsulfanyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(4-Bromo-phenylsulfanyl)-piperidine-1-carboxylic acid tert-butyl ester

4-(4-Bromo-phenylsulfanylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(4-Bromo-phenylsulfanylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-(4-Bromo-phenylsulfanylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

(R)-3-(4-Bromo-benzenesulfinyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(4-Bromo-benzenesulfinyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(4-Bromo-benzenesulfinyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(4-Bromo-benzenesulfinylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-(4-Bromo-benzenesulfinylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

(R)-3-(4-Bromo-benzenesulfinyl)-pyrrolidine

(S)-3-(4-Bromo-benzenesulfinyl)-pyrrolidine

3-(4-Bromo-benzenesulfinyl)-pyrrolidine

3-(4-Bromo-benzenesulfinylmethyl)-pyrrolidine

2-(4-Bromo-benzenesulfinylmethyl)-pyrrolidine

4-(4-Bromo-benzenesulfinyl)-piperidine

3-(4-Bromo-benzenesulfinyl)-piperidine

4-(4-Bromo-benzenesulfinylmethyl)-piperidine

3-(4-Bromo-benzenesulfinylmethyl)-piperidine

2-(4-Bromo-benzenesulfinylmethyl)-piperidine

4-(4-Bromo-benzenesulfinyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(4-Bromo-benzenesulfinyl)-piperidine-1-carboxylic acid tert-butyl ester

4-(4-Bromo-benzenesulfinylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(4-Bromo-benzenesulfinylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-(4-Bromo-benzenesulfinylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

(R)-3-(4-Bromo-benzenesulfonyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(4-Bromo-benzenesulfonyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(4-Bromo-benzenesulfonyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(4-Bromo-benzenesulfonylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-(4-Bromo-benzenesulfonylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

(R)-3-(4-Bromo-benzenesulfonyl)-pyrrolidine

(S)-3-(4-Bromo-benzenesulfonyl)-pyrrolidine

3-(4-Bromo-benzenesulfonyl)-pyrrolidine

3-(4-Bromo-benzenesulfonylmethyl)-pyrrolidine

2-(4-Bromo-benzenesulfonylmethyl)-pyrrolidine

4-(4-Bromo-benzenesulfonyl)-piperidine

3-(4-Bromo-benzenesulfonyl)-piperidine

4-(3-Cyano-pyridin-2-yl)-piperazine-1,3-dicarboxylic acid 1-tert-butylester

4-(4-Cyano-pyridin-2-yl)-3-methyl-piperazine-1-carboxylic acid tert-butyl ester

(4 -Cyano-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-yl)-methyl-carbamic acid tert-butyl ester

(4 -Cyano-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-yl)-methyl-carbamic acid tert-butyl ester

2-[(6-Bromo-pyridin-2-ylamino)-methyl]-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(6-Bromo-pyridin-2-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-Bromo-6-((S)-pyrrolidin-3-yloxy)-pyridine hydrochloride

(R)-3-(6-Bromo-pyridin-2-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-Bromo-6-((R)-pyrrolidin-3-yloxy)-pyridine hydrochloride

(S)-1-(6-Bromo-pyridin-2-yl)-pyrrolidin-3-ol

(R)-1-(6-Bromo-pyridin-2-yl)-pyrrolidin-3-ol

4-[(6-Bromo-pyridin-2-yl)-methyl-amino]-piperidine-1-carboxylic acid tert-butyl ester

2-(6-Bromo-pyridin-2-yloxymethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-[(6-Bromo-pyridin-2-yl)-methyl-amino]-piperidine-1-carboxylic acid tert-butyl ester

(6-Bromo-pyridin-2-yl)-methyl-piperidin-3-yl-amine hydrochloride

1-(4-Methyl-pyridin-2-yl)-pyrrolidin-3-ol

4-((S)-Pyrrolidin-3-yloxy)-pyridine hydrochloride

4-((R)-Pyrrolidin-3-yloxy)-pyridine hydrochloride

4-(Piperidin-3-ylmethoxy)-pyridine hydrochloride

4-(Piperidin-4-ylmethoxy)-pyridine hydrochloride

4-(6-Chloro-pyridin-3-ylmethyl)-piperazine-1,3-dicarboxylic acid 1-tert-butyl ester 3-(6-chloro-pyridin-3-ylmethyl) ester

1-(6-Chloro-pyridin-3-ylmethyl)-piperidine-2-carboxylic acid 6-chloro-pyridin-3-ylmethyl ester

1-(6-Ethoxy-pyridin-3-ylmethyl)-piperazine dihydrochloride

4-(Piperidin-3-yloxymethyl)-pyridine hydrochloride

2-(6-Chloro-pyridin-3-ylmethoxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-Chloro-5-(piperidin-2-ylmethoxymethyl)-pyridine hydrochloride

2-Chloro-5-(piperidin-4-ylmethoxymethyl)-pyridine hydrochloride

4-(6-Chloro-pyridin-3-ylmethyl)-piperazine-2-carboxylic acid

4-(6-Chloro-pyridin-3-ylmethyl)-piperazine-1,3-dicarboxylic acid 1-tert-butyl ester

1-(6-Chloro-pyridin-3-ylmethyl)-piperazine-2-carboxylic acid hydrochloride

1-(6-Chloro-pyridin-3-ylmethyl)-piperidine-2-carboxylic acid

1-(6-Bromo-pyridin-2-yl)-piperazine-2-carboxylic acid hydrochloride

2-(6-Bromo-pyridin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-Bromo-6-(piperidin-2-ylmethoxy)-pyridine hydrochloride

4-(6-Bromo-pyridin-2-yl)-piperazine-2-carboxylic acid

2-(5-Nitro-pyridin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-Nitro-2-(piperidin-2-ylmethoxy)-pyridine hydrochloride

4-(3-Nitro-pyridin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

4-(3-Nitro-pyridin-2-yl)-piperazine-2-carboxylic acid

4-(5-Nitro-pyridin-2-yl)-piperazine-1,3-dicarboxylic acid 1-tert-butylester

1-(5-Nitro-pyridin-2-yl)-piperazine-2-carboxylic acid hydrochloride

4-(3-Nitro-pyridin-2-yl)-piperazine-1,3-dicarboxylic acid 1-tert-butylester

1-(3-Nitro-pyridin-2-yl)-piperazine-2-carboxylic acid hydrochloride

2-(4-Cyano-pyridin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-(Piperidin-2-ylmethoxy)-isonicotinonitrile hydrochloride

2-(3-Cyano-pyridin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-(Piperidin-2-ylmethoxy)-nicotinonitrile hydrochloride

2-(Piperidin-4-ylmethoxy)-nicotinonitrile hydrochloride

4-(4-Cyano-pyridin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-(Piperidin-4-ylmethoxy)-isonicotinonitrile hydrochloride

4-(4-Cyano-pyridin-2-yl)-piperazine-2-carboxylic acid

4-(3-Cyano-pyridin-2-yl)-piperazine-2-carboxylic acid

4-(4-Cyano-pyridin-2-yl)-piperazine-1,3-dicarboxylic acid 1-tert-butylester

1-(4-Cyano-pyridin-2-yl)-piperazine-2-carboxylic acid hydrochloride

1-(3-Cyano-pyridin-2-yl)-piperazine-2-carboxylic acid hydrochloride

2-(Piperidin-4-ylmethoxymethyl)-pyridine hydrochloride

4-Pyridin-4-ylmethyl-piperazine-2-carboxylic acid

4-Pyridin-2-ylmethyl-piperazine-2-carboxylic acid

1-Pyridin-2-ylmethyl-piperazine-2-carboxylic acid hydrochloride

1-Pyridin-4-ylmethyl-piperazine-2-carboxylic acid hydrochloride

(6 -Bromo-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-2-yl)-methanol

4 -Methyl-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-2-carboxylic acid

4 -Methyl-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-carboxylic acid

(1r,4r)-N1-(pyridin-2-ylmethyl)cyclohexane-1,4-diamine hydrochloride

(1r,4r)-4-(pyridin-2-ylmethylamino)cyclohexanol

N-Pyridin-2-ylmethyl-cyclohexane-1,4-diamine hydrochloride

N-Pyridin-2-ylmethyl-cyclohexane-1,2-diamine hydrochloride

(1r,4r)-N1-(pyridin-4-ylmethyl)cyclohexane-1,4-diamine hydrochloride

(1r,4r)-4-(pyridin-4-ylmethylamino)cyclohexanol

N-Pyridin-4-ylmethyl-cyclohexane-1,4-diamine hydrochloride

N-Pyridin-4-ylmethyl-cyclohexane-1,2-diamine hydrochloride

{4-[(6-Chloro-pyridin-3-ylmethyl)-amino]-cyclohexyl}-carbamic acid tert-butyl ester

(1r,4r)-N1-((6-chloropyridin-3-yl)methyl)cyclohexane-1,4-diamine hydrochloride

N-(6-Chloro-pyridin-3-ylmethyl)-cyclohexane-1,4-diamine hydrochloride

{2-[(6-Chloro-pyridin-3-ylmethyl)-amino]-cyclohexyl}-carbamic acid tert-butyl ester

N-(6-Chloro-pyridin-3-ylmethyl)-cyclohexane-1,2-diamine hydrochloride

2-((1r,4r)-4-hydroxycyclohexylamino)isonicotinonitrile

2-((1r,4r)-4-hydroxycyclohexylamino)nicotinonitrile

[4-(3-Nitro-pyridin-2-ylamino)-cyclohexyl]-carbamic acid tert-butyl ester

(1r,4r)-N1-(3-nitropyridin-2-yl)cyclohexane-1,4-diamine hydrochloride

N-(3-Nitro-pyridin-2-yl)-cyclohexane-1,4-diamine hydrochloride

[2-(3-Nitro-pyridin-2-ylamino)-cyclohexyl]-carbamic acid tert-butyl ester

N-(3-Nitro-pyridin-2-yl)-cyclohexane-1,2-diamine hydrochloride

[4-(5-Nitro-pyridin-2-ylamino)-cyclohexyl]-carbamic acid tert-butyl ester

(1r,4r)-N1-(5-nitropyridin-2-yl)cyclohexane-1,4-diamin e hydrochloride

N-(5-Nitro-pyridin-2-yl)-cyclohexane-1,4-diamine hydrochloride

[2-(5-Nitro-pyridin-2-ylamino)-cyclohexyl]-carbamic acid tert-butyl ester

N-(5-Nitro-pyridin-2-yl)-cyclohexane-1,2-diamine hydrochloride

(1r,4r)-4-(5-methylpyridin-2-ylamino)cyclohexanol

(1r,4r)-4-(4-methylpyridin-2-ylamino)cyclohexanol

[4-(6-Bromo-pyridin-2-ylamino)-cyclohexyl]-carbamic acid tert-butyl ester

(1r,4r)-N1-(6-bromopyridin-2-yl)cyclohexane-1,4-diamine hydrochloride

(1r,4r)-4-(6-bromopyridin-2-ylamino)cyclohexanol

N-(6-Bromo-pyridin-2-yl)-cyclohexane-1,4-diamine hydrochloride

[2-(6-Bromo-pyridin-2-ylamino)-cyclohexyl]-carbamic acid tert-butyl ester

N-(6-Bromo-pyridin-2-yl)-cyclohexane-1,2-diamine hydrochloride

(1r,4r)-4-(pyridin-2-ylamino)cyclohexanol

(1r,4r)-4-(pyridin-4-ylamino)cyclohexanol

3-[(6-Chloro-pyridin-3-ylmethyl)-amino]-pyrrolidine-1-carboxylic acid tert-butyl ester

(6-Chloro-pyridin-3-ylmethyl)-pyrrolidin-3-yl-amine hydrochloride

(S)-3-[(6-Chloro-pyridin-3-ylmethyl)-amino]-pyrrolidine-1-carboxylic acid tert-butyl ester

(6-Chloro-pyridin-3-ylmethyl)-(S)-pyrrolidin-3-yl-amine hydrochloride

(R)-3-[(6-Chloro-pyridin-3-ylmethyl)-amino]-pyrrolidine-1-carboxylic acid tert-butyl ester

(6-Chloro-pyridin-3-ylmethyl)-(R)-pyrrolidin-3-yl-amine hydrochloride

(6-Chloro-pyridin-3-ylmethyl)-pyrrolidin-2-ylmethyl-amine hydrochloride

2-Chloro-5-((S)-pyrrolidin-3-yloxymethyl)-pyridine hydrochloride

1-(6-Chloro-pyridin-3-ylmethyl)-pyrrolidin-3-ol

(S)-1-(6-Chloro-pyridin-3-ylmethyl)-pyrrolidin-3-ol

(R)-1-(6-Chloro-pyridin-3-ylmethyl)-pyrrolidin-3-ol

1-(6-Chloro-pyridin-3-ylmethyl)-azetidine-3-carboxylic acid

[1-(6-Chloro-pyridin-3-ylmethyl)-piperidin-4-yl]-methyl-amine hydrochloride

2-Chloro-5-(pyrrolidin-2-ylmethoxymethyl)-pyridine hydrochloride

2-{[(6-Chloro-pyridin-3-ylmethyl)-amino]-methyl}-piperidine-1-carboxylic acid tert-butyl ester

(6-Chloro-pyridin-3-ylmethyl)-piperidin-2-ylmethyl-amine hydrochloride

2-(Pyrrolidin-3-ylamino)-isonicotinonitrile hydrochloride

(S)-3-(4-Cyano-pyridin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-((S)-Pyrrolidin-3-ylamino)-isonicotinonitrile hydrochloride

(R)-3-(4-Cyano-pyridin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-((R)-Pyrrolidin-3-ylamino)-isonicotinonitrile hydrochloride

2-[(4-Cyano-pyridin-2-ylamino)-methyl]-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(4-Cyano-pyridin-2-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-((S)-Pyrrolidin-3-yloxy)-isonicotinonitrile hydrochloride

(R)-3-(4-Cyano-pyridin-2-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-((R)-Pyrrolidin-3-yloxy)-isonicotinonitrile hydrochloride

1-(4-Cyano-pyridin-2-yl)-azetidine-3-carboxylic acid

2-(2-Methyl-piperazin-1-yl)-isonicotinonitrile hydrochloride

4-(4-Cyano-pyridin-2-yl)-2-methyl-piperazine-1-carboxylic acid tert-butyl ester

2-(3-Methyl-piperazin-1-yl)-isonicotinonitrile hydrochloride

4-Methylamino-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4 -carbonitrile hydrochloride

2-(4-Cyano-pyridin-2-yloxymethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-(Pyrrolidin-2-ylmethoxy)-isonicotinonitrile hydrochloride

3-[(4-Cyano-pyridin-2-yl)-methyl-amino]-piperidine-1-carboxylic acid tert-butyl ester

2-(Methyl-piperidin-3-yl-amino)-isonicotinonitrile hydrochloride

3-Methylamino-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4 -carbonitrile hydrochloride

3-(6-Bromo-pyridin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butylester

(6-Bromo-pyridin-2-yl)-pyrrolidin-3-yl-amine hydrochloride

(S)-3-(6-Bromo-pyridin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

(6-Bromo-pyridin-2-yl)-(S)-pyrrolidin-3-yl-amine hydrochloride

(R)-3-(6-Bromo-pyridin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

(6-Bromo-pyridin-2-yl)-(R)-pyrrolidin-3-yl-amine hydrochloride

(6-Bromo-pyridin-2-yl)-pyrrolidin-2-ylmethyl-amine hydrochloride

1-(6-Bromo-pyridin-2-yl)-azetidine-3-carboxylic acid

4-(6-Bromo-pyridin-2-yl)-[1,4]diazepane-1-carboxylic acid tert-butyl ester

1-(6-Bromo-pyridin-2-yl)-[1,4]diazepane hydrochloride

4-(6-Bromo-pyridin-2-yl)-3-methyl-piperazine-1-carboxylic acid tert-butyl ester

1-(6-Bromo-pyridin-2-yl)-2-methyl-piperazine hydrochloride

4-(6-Bromo-pyridin-2-yl)-2-methyl-piperazine-1-carboxylic acid tert-butyl ester

1-(6-Bromo-pyridin-2-yl)-3-methyl-piperazine hydrochloride

(6 -Bromo-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-yl)-methyl-carbamic acid tert-butyl ester

(6 -Bromo-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-4-yl)-methyl-amine hydrochloride

(6-Bromo-pyridin-2-yl)-methyl-piperidin-4-yl-amine hydrochloride

2-Bromo-6-(pyrrolidin-2-ylmethoxy)-pyridine hydrochloride

2-[(6-Bromo-pyridin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

(6-Bromo-pyridin-2-yl)-piperidin-2-ylmethyl-amine hydrochloride

(6 -Bromo-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-yl)-methyl-carbamic acid tert-butyl ester

(6 -Bromo-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-yl)-methyl-amine hydrochloride

3-(4-Methyl-pyridin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

(4-Methyl-pyridin-2-yl)-pyrrolidin-3-yl-amine hydrochloride

(S)-3-(4-Methyl-pyridin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

(4-Methyl-pyridin-2-yl)-(S)-pyrrolidin-3-yl-amine hydrochloride

(R)-3-(4-Methyl-pyridin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

(4-Methyl-pyridin-2-yl)-(R)-pyrrolidin-3-yl-amine hydrochloride

2-[(4-Methyl-pyridin-2-ylamino)-methyl]-pyrrolidine-1-carboxylic acid tert-butyl ester

(4-Methyl-pyridin-2-yl)-pyrrolidin-2-ylmethyl-amine hydrochloride

(S)-3-(4-Methyl-pyridin-2-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

4-Methyl-2-((S)-pyrrolidin-3-yloxy)-pyridine hydrochloride

(R)-3-(4-Methyl-pyridin-2-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

4-Methyl-2-((R)-pyrrolidin-3-yloxy)-pyridine hydrochloride

(S)-1-(4-Methyl-pyridin-2-yl)-pyrrolidin-3-ol

(R)-1-(4-Methyl-pyridin-2-yl)-pyrrolidin-3-ol

3-Methyl-4-(4-methyl-pyridin-2-yl)-piperazine-1-carboxylic acid tert-butyl ester

2-Methyl-1-(4-methyl-pyridin-2-yl)-piperazine hydrochloride

2-Methyl-4-(4-methyl-pyridin-2-yl)-piperazine-1-carboxylic acid tert-butyl ester

3-Methyl-1-(4-methyl-pyridin-2-yl)-piperazine hydrochloride

4-[Methyl-(4-methyl-pyridin-2-yl)-amino]-piperidine-1-carboxylic acid tert-butyl ester

Methyl-(4-methyl-pyridin-2-yl)-piperidin-4-yl-amine hydrochloride

3-[Methyl-(4-methyl-pyridin-2-yl)-amino]-piperidine-1-carboxylic acid tert-butyl ester

Methyl-(4-methyl-pyridin-2-yl)-piperidin-3-yl-amine hydrochloride

Methyl-(4 -methyl-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-yl)-carbamic acid tert-butyl ester

Methyl-(4 -methyl-3,4,5,6-tetrahydro-2H-[1,2 ]bipyridinyl-3-yl)-amine hydrochloride

Methyl-piperidin-3-yl-pyridin-4-yl-amine hydrochloride

(R)-3-(Pyridin-4-ylsulfanyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(Pyridin-4-ylsulfanyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(Pyridin-4-ylsulfanyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(Pyridin-4-ylsulfanylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-(Pyridin-4-ylsulfanylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

4-((R)-Pyrrolidin-3-ylsulfanyl)-pyridine

4-((S)-Pyrrolidin-3-ylsulfanyl)-pyridine

4-(Pyrrolidin-3-ylsulfanyl)-pyridine

4-(Pyrrolidin-3-ylmethylsulfanyl)-pyridine

4-(Pyrrolidin-2-ylmethylsulfanyl)-pyridine

4-(Piperidin-4-ylsulfanyl)-pyridine

4-(Piperidin-3-ylsulfanyl)-pyridine

4-(Piperidin-4-ylmethylsulfanyl)-pyridine

4-(Piperidin-3-ylmethylsulfanyl)-pyridine

4-(Piperidin-2-ylmethylsulfanyl)-pyridine

4-(Pyridin-4-ylsulfanyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(Pyridin-4-ylsulfanyl)-piperidine-1-carboxylic acid tert-butyl ester

4-(Pyridin-4-ylsulfanylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(Pyridin-4-ylsulfanylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-(Pyridin-4-ylsulfanylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

(R)-3-(Pyridine-4-sulfinyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(Pyridine-4-sulfinyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(Pyridine-4-sulfinyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(Pyridine-4-sulfinylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-(Pyridine-4-sulfinylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

4-((R)-Pyrrolidine-3-sulfinyl)-pyridine

4-((S)-Pyrrolidine-3-sulfinyl)-pyridine

4-(Pyrrolidine-3-sulfinyl)-pyridine

4-(Pyrrolidin-3-ylmethanesulfinyl)-pyridine

4-(Pyrrolidin-2-ylmethanesulfinyl)-pyridine

4-(Piperidine-4-sulfinyl)-pyridine

4-(Piperidine-3-sulfinyl)-pyridine

4-(Piperidin-4-ylmethanesulfinyl)-pyridine

4-(Piperidin-3-ylmethanesulfinyl)-pyridine

4-(Piperidin-2-ylmethanesulfinyl)-pyridine

4-(Pyridine-4-sulfinyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(Pyridine-4-sulfinyl)-piperidine-1-carboxylic acid tert-butyl ester

4-(Pyridine-4-sulfinylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(Pyridine-4-sulfinylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-(Pyridine-4-sulfinylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

(R)-3-(Pyridine-4-sulfonyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(Pyridine-4-sulfonyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(Pyridine-4-sulfonyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(Pyridine-4-sulfonylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-(Pyridine-4-sulfonylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

4-((R)-Pyrrolidine-3-sulfonyl)-pyridine

4-((S)-Pyrrolidine-3-sulfonyl)-pyridine

4-(Pyrrolidine-3-sulfonyl)-pyridine

4-(Pyrrolidin-3-ylmethanesulfonyl)-pyridine

4-(Pyrrolidin-2-ylmethanesulfonyl)-pyridine

4-(Piperidine-4-sulfonyl)-pyridine

4-(Piperidine-3-sulfonyl)-pyridine

4-(Piperidin-4-ylmethanesulfonyl)-pyridine

4-(Piperidin-3-ylmethanesulfonyl)-pyridine

4-(Piperidin-2-ylmethanesulfonyl)-pyridine

4-(Pyridine-4-sulfonyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(Pyridine-4-sulfonyl)-piperidine-1-carboxylic acid tert-butyl ester

4-(Pyridine-4-sulfonylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(Pyridine-4-sulfonylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-(Pyridine-4-sulfonylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

(R)-3-(Pyridin-2-ylsulfanyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(Pyridin-2-ylsulfanyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(Pyridin-2-ylsulfanyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(Pyridin-2-ylsulfanylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-(Pyridin-2-ylsulfanylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-((R)-Pyrrolidin-3-ylsulfanyl)-pyridine

2-((S)-Pyrrolidin-3-ylsulfanyl)-pyridine

2-(Pyrrolidin-3-ylsulfanyl)-pyridine

2-(Pyrrolidin-3-ylmethylsulfanyl)-pyridine2-(Pyrrolidin-3-ylmethylsulfanyl)-pyridine

2-(Pyrrolidin-2-ylmethylsulfanyl)-pyridine

2-(Piperidin-4-ylsulfanyl)-pyridine

2-(Piperidin-3-ylsulfanyl)-pyridine

2-(Piperidin-4-ylmethylsulfanyl)-pyridine

2-(Piperidin-3-ylmethylsulfanyl)-pyridine

2-(Piperidin-2-ylmethylsulfanyl)-pyridine

4-(Pyridin-2-ylsulfanyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(Pyridin-2-ylsulfanyl)-piperidine-1-carboxylic acid tert-butyl ester

4-(Pyridin-2-ylsulfanylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(Pyridin-2-ylsulfanylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-(Pyridin-2-ylsulfanylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

(R)-3-(Pyridine-2-sulfinyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(Pyridine-2-sulfinyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(Pyridine-2-sulfinyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(Pyridine-2-sulfinylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-(Pyridine-2-sulfinylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-((R)-Pyrrolidine-3-sulfinyl)-pyridine

2-((S)-Pyrrolidine-3-sulfinyl)-pyridine

2-(Pyrrolidine-3-sulfinyl)-pyridine

2-(Pyrrolidin-3-ylmethanesulfinyl)-pyridine

2-(Pyrrolidin-2-ylmethanesulfinyl)-pyridine

2-(Piperidine-4-sulfinyl)-pyridine

2-(Piperidine-3-sulfinyl)-pyridine

2-(Piperidin-4-ylmethanesulfinyl)-pyridine

2-(Piperidin-3-ylmethanesulfinyl)-pyridine

2-(Piperidin-2-ylmethanesulfinyl)-pyridine

4-(Pyridine-2-sulfinyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(Pyridine-2-sulfinyl)-piperidine-1-carboxylic acid tert-butyl ester

4-(Pyridine-2-sulfinylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(Pyridine-2-sulfinylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-(Pyridine-2-sulfinylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

(R)-3-(Pyridine-2-sulfonyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(Pyridine-2-sulfonyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(Pyridine-2-sulfonyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(Pyridine-2-sulfonylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-(Pyridine-2-sulfonylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-((R)-Pyrrolidine-3-sulfonyl)-pyridine

2-((S)-Pyrrolidine-3-sulfonyl)-pyridine

2-(Pyrrolidine-3-sulfonyl)-pyridine

2-(Pyrrolidin-3-ylmethanesulfonyl)-pyridine

2-(Pyrrolidin-2-ylmethanesulfonyl)-pyridine

2-(Piperidine-4-sulfonyl)- pyridine

2-(Piperidine-3-sulfonyl)- pyridine

2-(Piperidin-4-ylmethanesulfonyl)-pyridine

2-(Piperidin-3-ylmethanesulfonyl)-pyridine

2-(Piperidin-2-ylmethanesulfonyl)-pyridine

4-(Pyridine-2-sulfonyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(Pyridine-2-sulfonyl)-piperidine-1-carboxylic acid tert-butyl ester

4-(Pyridine-2-sulfonylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(Pyridine-2-sulfonylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-(Pyridine-2-sulfonylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-(3-(chloromethyl)piperidin-1-yl)pyrimidine

N-cyclopropyl-6-(piperidin-4-yloxy)pyrimidin-4-amine hydrochloride

1-(6-Cyclopropylamino-pyrimidin-4-yl)-piperidin-4-ol

[6-(4-Amino-piperidin-1-yl)-pyrimidin-4-yl]-cyclopropyl-amine hydrochloride

Cyclopropyl-(6-piperazin-1-yl-pyrimidin-4-yl)-amine hydrochloride

N,N-Dimethyl-N -piperidin-4-yl-pyrimidine-4,6-diamine hydrochloride

N,N-dimethyl-6-(piperazin-1-yl)pyrimidin-4-amine hydrochloride

1-(6-Ethoxy-pyrimidin-4-yl)-piperidin-3-ol

1-(6-Ethoxy-pyrimidin-4-yl)-piperidin-3-ylamine hydrochloride

[6-(3-Amino-piperidin-1-yl)-pyrimidin-4-yl]-diethyl-amine hydrochloride

1-(6-Diethylamino-pyrimidin-4-yl)-piperidin-4-ol

1-(6-Diethylamino-pyrimidin-4-yl)-piperidin-3-ol

Diethyl-(6-piperazin-1-yl-pyrimidin-4-yl)-amine hydrochloride

[6-(4-Amino-piperidin-1-yl)-pyrimidin-4-yl]-diethyl-amine hydrochloride

1-(6-Methoxy-pyrimidin-4-yl)-piperidin-4-ylamine hydrochloride

4-Methoxy-6-piperazin-1-yl-pyrimidine hydrochloride

1-(6-Methoxy-pyrimidin-4-yl)-piperidin-3-ylamine hydrochloride

1-(6-Methoxy-pyrimidin-4-yl)-piperidin-4-ol

1-(6-Methoxy-pyrimidin-4-yl)-piperidin-3-ol

2-(Piperidin-4-yloxy)-pyrimidine hydrochloride

2-(Piperidin-3-yloxy)-pyrimidine hydrochloride

2-(Piperidin-3-ylmethoxy)-pyrimidine hydrochloride

(6-Chloro-pyrimidin-4-yl)-piperidin-4-yl-amine hydrochloride

1-Pyrimidin-2-yl-piperidin-3-ol

1-Pyrimidin-2-yl-piperidine-4-carboxylic acid

(1-Pyrimidin-2-yl-piperidin-3-yl)-methanol

Piperidin-3-ylmethyl-pyrimidin-2-yl-amine hydrochloride

Piperidin-3-yl-pyrimidin-2-yl-amine hydrochloride

Piperidin-4-yl-pyrimidin-2-yl-amine hydrochloride

Piperidin-4-ylmethyl-pyrimidin-2-yl-amine hydrochloride

4-(6-Chloro-pyrimidin-4-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

(6-Chloro-pyrimidin-4-yl)-piperidin-4-ylmethyl-amine hydrochloride

Quinoxalin-2-yl-piperidin-4-ol

4-[(6-Chloro-pyrimidin-4-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

(6-Chloro-pyrimidin-4-yl)-piperidin-3-yl-amine hydrochloride

Quinoxalin-2-yl-piperidin-3-ol

3-(6-Chloro-pyrimidin-4-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

(6-Chloro-pyrimidin-4-yl)-piperidin-3-ylmethyl-amine hydrochloride

3-[(6-Chloro-pyrimidin-4-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

(1-Quinoxalin-2-yl-piperidin-3-yl)-Methanol

1-(3-Cyclopropylamino-quinoxalin-2-yl)-piperidin-4-ol

(3-Chloro-quinoxalin-2-yl)-cyclopropyl-amine

Piperidin-4-yl-quinoxalin-2-yl-amine hydrochloride

Piperidin-4-ylmethyl-quinoxalin-2-yl-amine hydrochloride

2-Piperazin-1-yl-quinoxaline hydrochloride

4-Chloro-6-(piperidin-4-yloxy)-pyrimidine hydrochloride

1-Quinoxalin-2-yl-piperidin-4-ylamine hydrochloride

[3-(4-Amino-piperidin-1-yl)-quinoxalin-2-yl]-cyclopropyl-amine hydrochloride

Cyclopropyl-(3-piperazin-1-yl-quinoxalin-2-yl)-amine hydrochloride

N-Cyclopropyl-N -piperidin-4-yl-quinoxaline-2,3-diamine hydrochloride

Piperidin-3-ylmethyl-quinoxalin-2-yl-amine hydrochloride

2-(piperidin-4-yloxy)quinoxaline hydrochloride

2-(piperidin-3-ylmethoxy)quinoxaline hydrochloride

tert-butyl-4-(3-(cyclopropylamino)quinoxalin-2-yloxy)piperidine-1-carboxylate

2-(6-Bromo-pyridin-2-yloxy)-quinoxaline

2-(4-Chloro-pyrimidin-2-yloxy)-quinoxaline

2-(6-Chloro-pyrimidin-4-yloxy)-quinoxaline

2-(6-Chloro-pyridazin-3-yloxy)-quinoxaline

2-(5-Chloromethyl-thiazol-2-yloxy)-quinoxaline

3-(3-Methoxy-quinoxalin-2-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

3-[(3-Methoxy-quinoxalin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

4-[(3-Methoxy-quinoxalin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

2-(5-Chloromethyl-pyridin-2-yloxy)-quinoxaline

4-(3-Methoxy-quinoxalin-2-yl)-piperazine-1-carboxylic acid tert-butyl ester

[1-(3-Methoxy-quinoxalin-2-yl)-piperidin-4-yl]-carbamic acid tert-butyl ester

[1-(3-Methoxy-quinoxalin-2-yl)-piperidin-3-yl]-carbamic acid tert-butyl ester

1-(3-Methoxy-quinoxalin-2-yl)-piperidin-4-ol

4-Chloro-6-(piperidin-3-yloxy)-pyrimidine hydrochloride

3-(6-Chloro-pyrimidin-4-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

1-(6-Chloro-pyrimidin-4-yl)-piperidin-4-ylamine hydrochloride

(3-Chloro-quinoxalin-2-yl)-piperidin-4-yl-amine hydrochloride

[1-(6-Chloro-pyrimidin-4-yl)-piperidin-4-yl]-carbamic acid tert-butyl ester

1-(6-Chloro-pyrimidin-4-yl)-piperidin-3-ylamine hydrochloride

[1-(6-Chloro-pyrimidin-4-yl)-piperidin-3-yl]-carbamic acid tert-butyl ester

4-(3-Chloro-quinoxalin-2-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

4-Chloro-6-piperazin-1-yl-pyrimidine hydrochloride

4-(6-Chloro-pyrimidin-4-yl)-piperazine-1-carboxylic acid tert-butyl ester

(3-Chloro-quinoxalin-2-yl)-piperidin-4-ylmethyl-amine hydrochloride

1-(6-Chloro-pyrimidin-4-yl)-piperidine-4-carboxylic acid

2-(1-piperazinyl)-pyrimidine hydrochloride

4-[(3-Chloro-quinoxalin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

1-(2-pyrimidinyl)-4-piperidinamine hydrochloride

1-(6-Chloro-pyrimidin-4-yl)-piperidin-4-ol

1-(6-Chloro-pyrimidin-4-yl)-piperidin-3-ol

[1-(6-Chloro-pyrimidin-4-yl)-piperidin-3-yl]-methanol

(3-Chloro-quinoxalin-2-yl)-piperidin-3-yl-amine hydrochloride

1-Pyrimidin-2-yl-piperidin-4-ol

1-(2-pyrimidinyl)-3-piperidinamine hydrochloride

3-(3-Chloro-quinoxalin-2-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

[1-(4-Trifluoromethyl-pyrimidin-2-yl)-piperidin-3-yl]-methanol

1-(4-Trifluoromethyl-pyrimidin-2-yl)-piperidin-4-ol

2-(5-Chloro-pyrimidin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(5-Chloro-pyrimidin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

(3-Chloro-quinoxalin-2-yl)-piperidin-3-ylmethyl-amine hydrochloride

4-(5-Chloro-pyrimidin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

4-(5-Chloro-pyrimidin-2-yloxy)-piperidine-1-carboxylic acid tert-butylester

3-[(3-Chloro-quinoxalin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

4-(5-Chloro-pyrimidin-2-yl)-piperazine-1,3-dicarboxylic acid 1-tert-butyl ester

[1-(5-Chloro-pyrimidin-2-yl)-piperidin-2-yl]-methanol

[1-(5-Chloro-pyrimidin-2-yl)-piperidin-3-yl]-methanol

[1-(5-Chloro-pyrimidin-2-yl)-piperidin-4-yl]-methanol

1-(5-Chloro-pyrimidin-2-yl)-piperidine-2-carboxylic acid

1-(5-Chloro-pyrimidin-2-yl)-piperidine-3-carboxylic acid

4-(3-Chloro-quinoxalin-2-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

1-(5-Chloro-pyrimidin-2-yl)-piperidine-4-carboxylic acid

1-(5-Chloro-pyrimidin-2-yl)-piperidin-3-ol

1-(5-Chloro-pyrimidin-2-yl)-piperidin-4-ol

3-(5-Chloro-pyrimidin-2-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

(5-Chloro-pyrimidin-2-yl)-piperidin-3-yl-amine hydrochloride

3-(3-Chloro-quinoxalin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(3-Chloro-quinoxalin-2-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

4-(5-Chloro-pyrimidin-2-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

(5-Chloro-pyrimidin-2-yl)-piperidin-4-yl-amine hydrochloride

1-(3-Chloro-quinoxalin-2-yl)-piperidin-4-ylamine hydrochloride

[1-(3-Chloro-quinoxalin-2-yl)-piperidin-4-yl]-carbamic acid tert-butyl ester

1-(3-Chloro-quinoxalin-2-yl)-piperidin-3-ylamine hydrochloride

[1-(3-Chloro-quinoxalin-2-yl)-piperidin-3-yl]-carbamic acid tert-butyl ester

[1-(5-Chloro-pyrimidin-2-yl)-piperidin-4-yl]-carbamic acid tert-butyl ester

2-Chloro-3-piperazin-1-yl-quinoxaline hydrochloride

2-(4,6-Dimethyl-pyrimidin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(4,6-Dimethyl-pyrimidin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(4,6-Dimethyl-pyrimidin-2-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

4-(3-Chloro-quinoxalin-2-yl)-piperazine-1-carboxylic acid tert-butyl ester

4-(4,6-Dimethyl-pyrimidin-2-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

1-(3-Chloro-quinoxalin-2-yl)-piperidine-4-carboxylic acid

4-(4,6-Dimethyl-pyrimidin-2-yl)-piperazine-1,3-dicarboxylic acid 1-tert-butyl ester

2-(5-Fluoro-pyrimidin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

1-(3-Chloro-quinoxalin-2-yl)-piperidin-4-ol

3-(5-Fluoro-pyrimidin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

1-(3-Chloro-quinoxalin-2-yl)-piperidin-3-ol

4-(5-Fluoro-pyrimidin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(5-Fluoro-pyrimidin-2-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

[1-(3-Chloro-quinoxalin-2-yl)-piperidin-3-yl]-methanol

4-(5-Fluoro-pyrimidin-2-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

1-(3-Chloro-quinoxalin-2-yl)-piperidine-3-carboxylic acid

4-(5-Fluoro-pyrimidin-2-yl)-piperazine-1,3-dicarboxylic acid 1-tert-butyl ester

[1-(5-Fluoro-pyrimidin-2-yl)-piperidin-3-yl]-methanol

[1-(3-Chloro-quinoxalin-2-yl)-piperidin-2-yl]-methanol

[1-(5-Fluoro-pyrimidin-2-yl)-piperidin-4-yl]-methanol

1-(5-Fluoro-pyrimidin-2-yl)-piperidine-2-carboxylic acid

[1-(3-Chloro-quinoxalin-2-yl)-piperidin-4-yl]-methanol

1-(5-Fluoro-pyrimidin-2-yl)-piperidine-3-carboxylic acid

1-(5-Fluoro-pyrimidin-2-yl)-piperidine-4-carboxylic acid

1-(5-Fluoro-pyrimidin-2-yl)-piperidin-3-ol

1-(5-Fluoro-pyrimidin-2-yl)-piperidin-4-ol

(5-Fluoro-pyrimidin-2-yl)-piperidin-3-yl-amine hydrochloride

4-(3-Chloro-quinoxalin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

4-(5-Fluoro-pyrimidin-2-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

(5-Fluoro-pyrimidin-2-yl)-piperidin-4-yl-amine hydrochloride

4-(3-Chloro-quinoxalin-2-yl)-piperazine-2-carboxylic acid

[1-(5-Fluoro-pyrimidin-2-yl)-piperidin-4-yl]-carbamic acid tert-butyl ester

4-(3-Chloro-quinoxalin-2-yl)-piperazine-1,3-dicarboxylic acid 1-tert-butyl ester

4-Pyrimidin-2-yl-piperazine-1,3-dicarboxylic acid 1-tert-butyl ester

1-(3-Chloro-quinoxalin-2-yl)-piperazine-2-carboxylic acid hydrochloride

3-(4-Methyl-pyrimidin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

(R)-3-(4-Methyl-pyrimidin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

1-(3-Chloro-quinoxalin-2-yl)-piperidine-2-carboxylic acid

(S)-3-(4-Methyl-pyrimidin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

1-(1-Thiazol-2-yl-ethyl)-piperazine hydrochloride

1-(1-Thiazol-2-yl-ethyl)-piperidin-4-ylamine hydrochloride

2-[(4-Methyl-pyrimidin-2-ylamino)-methyl]-pyrrolidine-1-carboxylic acid tert-butyl ester

(R)-3-(4-Methyl-pyrimidin-2-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(4-Methyl-pyrimidin-2-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-(4-Methyl-pyrimidin-2-yloxymethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

1-(4-Methyl-pyrimidin-2-yl)-pyrrolidin-3-ol

1-(1-Thiazol-2-yl-ethyl)-piperidin-4-ol

(R)-1-(4-Methyl-pyrimidin-2-yl)-pyrrolidin-3-ol

(S)-1-(4-Methyl-pyrimidin-2-yl)-pyrrolidin-3-ol

[1-(1-Thiazol-2-yl-ethyl)-piperidin-3-yl]-methanol

2-Methyl-4-(4-methyl-pyrimidin-2-yl)-piperazine-1-carboxylic acid tert-butyl ester

1-(4-Methyl-pyrimidin-2-yl)-piperidine-3-carboxylic acid

5-Chloromethyl-2-(furan-2-ylmethoxy)-thiazole

1-(4-Methyl-pyrimidin-2-yl)-piperidin-3-ol

2-Chloro-N-(1-thiazol-2-yl-piperidin-4-yl)-acetamide

1-(4-Methyl-pyrimidin-2-yl)-piperidin-4-ol

[1-(4-Methyl-pyrimidin-2-yl)-piperidin-2-yl]-methanol

2-Chloro-N-(1-thiazol-2-yl-piperidin-3-yl)-acetamide

[1-(4-Methyl-pyrimidin-2-yl)-piperidin-3-yl]-methanol

4-(Thiazol-2-yloxy)-piperidine hydrochloride

3-(Thiazol-2-yloxy)-piperidine hydrochloride

2-(3-Chloro-quinoxalin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

[1-(4-Methyl-pyrimidin-2-yl)-piperidin-4-yl]-methanol

2-Chloro-3-(piperidin-2-ylmethoxy)-quinoxaline hydrochloride

3-(Thiazol-2-yloxymethyl)-piperidine hydrochloride

2-Chloro-3-(piperidin-4-ylmethoxy)-quinoxaline hydrochloride

4-Thiazol-2-yl-morpholine

[1-(4-Methyl-pyrimidin-2-yl)-piperidin-3-yl]-carbamic acid tert-butyl ester

[4-(3-Chloro-quinoxalin-2-ylamino)-cyclohexyl]-carbamic acid tert-butyl ester

[1-(4-Methyl-pyrimidin-2-yl)-piperidin-4-yl]-carbamic acid tert-butyl ester

(1r,4r)-N1-(3-chloroquinoxalin-2-yl)cyclohexane-1,4-diamine hydrochloride

Methyl-[1-(4-methyl-pyrimidin-2-yl)-piperidin-4-yl]-carbamic acid tert-butyl ester

(1r,4r)-4-(3-chloroquinoxalin-2-ylamino)cyclohexanol

[1-(4-Methyl-pyrimidin-2-yl)-piperidin-4-ylmethyl]-carbamic acid tert-butyl ester

N-(3-Chloro-quinoxalin-2-yl)-cyclohexane-1,4-diamine hydrochloride

1-Thiazol-2-yl-piperidine

[2-(3-Chloro-quinoxalin-2-ylamino)-cyclohexyl]-carbamic acid tert-butyl ester

4-(2-Chloro-thiazol-5-ylmethoxy)-piperidine dihydrochloride

Methyl-[1-(4-methyl-pyrimidin-2-yl)-piperidin-3-yl]-carbamic acid tert-butyl ester

N-(3-Chloro-quinoxalin-2-yl)-cyclohexane-1,2-diamine hydrochloride

(1r,4r)-N1-(quinoxalin-2-yl)cyclohexane-1,4-diamine hydrochloride

3-(4-Methyl-pyrimidin-2-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

1-(2-thiazolyl)-piperazine hydrochloride

4-(4-Methyl-pyrimidin-2-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

(1r,4r)-4-(quinoxalin-2-ylamino)cyclohexanol

1-(2-thiazolyl)-3-piperidinamine hydrochloride

2-[(4-Methyl-pyrimidin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

N-Quinoxalin-2-yl-cyclohexane-1,4-diamine hydrochloride

3-[(4-Methyl-pyrimidin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

N-Quinoxalin-2-yl-cyclohexane-1,2-diamine hydrochloride

4-[(4-Methyl-pyrimidin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

3-[Methyl-(4-methyl-pyrimidin-2-yl)-amino]-piperidine-1-carboxylic acid tert-butyl ester

4-[Methyl-(4-methyl-pyrimidin-2-yl)-amino]-piperidine-1-carboxylic acid tert-butyl ester

3-(4-Methyl-pyrimidin-2-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

4-(4-Methyl-pyrimidin-2-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

2-(4-Methyl-pyrimidin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(4-Methyl-pyrimidin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

4-(4-Methyl-pyrimidin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(4-Chloro-5-methyl-pyrimidin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

(R)-3-(4-Chloro-5-methyl-pyrimidin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(4-Chloro-5-methyl-pyrimidin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-[(4-Chloro-5-methyl-pyrimidin-2-ylamino)-methyl]-pyrrolidine-1-carboxylic acid tert-butyl ester

(R)-3-(4-Chloro-5-methyl-pyrimidin-2-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(4-Chloro-5-methyl-pyrimidin-2-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

1-(4-Chloro-5-methyl-pyrimidin-2-yl)-pyrrolidin-3-ol

(R)-1-(4-Chloro-5-methyl-pyrimidin-2-yl)-pyrrolidin-3-ol

(S)-1-(4-Chloro-5-methyl-pyrimidin-2-yl)-pyrrolidin-3-ol

4-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperazine-1-carboxylic acid tert-butyl ester

4-Chloro-5-methyl-2-piperazin-1-yl-pyrimidine hydrochloride

4-(4-Chloro-5-methyl-pyrimidin-2-yl)-3-methyl-piperazine-1-carboxylic acid tert-butyl ester

4-Chloro-5-methyl-2-(2-methyl-piperazin-1-yl)-pyrimidine hydrochloride

4-(4-Chloro-5-methyl-pyrimidin-2-yl)-2-methyl-piperazine-1-carboxylic acid tert-butyl ester

4-Chloro-5-methyl-2-(3-methyl-piperazin-1-yl)-pyrimidine hydrochloride

4-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperazine-1,3-dicarboxylic acid 1-tert-butyl ester

1-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidine-2-carboxylic acid

1-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidine-3-carboxylic acid

1-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidine-4-carboxylic acid

1-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidin-3-ol

1-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidin-4-ol

[1-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidin-2-yl]-methanol

[1-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidin-3-yl]-methanol

[1-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidin-4-yl]-methanol

[1-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidin-3-yl]-carbamic acid tert-butyl ester

1-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidin-3-ylamine hydrochloride

[1-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidin-4-yl]-carbamic acid tert-butyl ester

[1-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidin-4-yl]-methyl-carbamic acid tert-butyl ester

[1-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidin-4-yl]-methyl-amine hydrochloride

[1-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidin-3-ylmethyl]-carbamic acid tert-butyl ester

[1-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidin-2-ylmethyl]-carbamic acid tert-butyl ester

[1-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidin-4-ylmethyl]-carbamic acid tert-butyl ester

C-[1-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidin-4-yl]-methylamine hydrochloride

[1-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidin-3-yl]-methyl-amine hydrochloride

3-(4-Chloro-5-methyl-pyrimidin-2-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

4-(4-Chloro-5-methyl-pyrimidin-2-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

2-[(4-Chloro-5-methyl-pyrimidin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

3-[(4-Chloro-5-methyl-pyrimidin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

4-[(4-Chloro-5-methyl-pyrimidin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidin-4-ylmethyl-amine hydrochloride

2-Chloro-N-(5-nitro-thiazol-2-yl)-acetamide

3-[(4-Chloro-5-methyl-pyrimidin-2-yl)-methyl-amino]-piperidine-1-carboxylic acid tert-butyl ester

4-[(4-Chloro-5-methyl-pyrimidin-2-yl)-methyl-amino]-piperidine-1-carboxylic acid tert-butyl ester

3-(4-Chloro-5-methyl-pyrimidin-2-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

4-(4-Chloro-5-methyl-pyrimidin-2-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

4-(4-Chloro-5-methyl-pyrimidin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(4-Chloro-6-methyl-pyrimidin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(4-Chloro-6-methyl-pyrimidin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

1-(4-Chloro-6-methyl-pyrimidin-2-yl)-pyrrolidin-3-ol

(R)-1-(4-Chloro-6-methyl-pyrimidin-2-yl)-pyrrolidin-3-ol

1-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidine-3-carboxylic acid

1-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidin-3-ol

[1-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidin-2-yl]-methanol

[1-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidin-3-yl]-methanol

[1-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidin-4-yl]-methanol

[1-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidin-4-yl]-carbamic acid tert-butyl ester

[1-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidin-4-ylmethyl]-carbamic acid tert-butyl ester

[1-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidin-3-yl]-methyl-carbamic acid tert-butyl ester

3-[(4-Chloro-6-methyl-pyrimidin-2-yl)-methyl-amino]-piperidine-1-carboxylic acid tert-butyl ester

(R)-3-(2-Chloro-6-methyl-pyrimidin-4-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(2-Chloro-6-methyl-pyrimidin-4-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-[(2-Chloro-6-methyl-pyrimidin-4-ylamino)-methyl]-pyrrolidine-1-carboxylic acid tert-butyl ester

1-(2-Chloro-6-methyl-pyrimidin-4-yl)-pyrrolidin-3-ol

(R)-1-(2-Chloro-6-methyl-pyrimidin-4-yl)-pyrrolidin-3-ol

(S)-1-(2-Chloro-6-methyl-pyrimidin-4-yl)-pyrrolidin-3-ol

4-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperazine-1-carboxylic acid tert-butyl ester

4-(2-Chloro-6-methyl-pyrimidin-4-yl)-3-methyl-piperazine-1-carboxylic acid tert-butyl ester

4-(2-Chloro-6-methyl-pyrimidin-4-yl)-2-methyl-piperazine-1-carboxylic acid tert-butyl ester

4-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperazine-1,3-dicarboxylic acid 1-tert-butyl ester

1-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidine-3-carboxylic acid

1-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-4-ol

[1-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-3-yl]-methanol

[1-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-4-yl]-carbamic acid tert-butyl ester

[1-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-4-yl]-methyl-carbamic acid tert-butyl ester

[1-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-2-ylmethyl]-carbamic acid tert-butyl ester

[1-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-3-ylmethyl]-carbamic acid tert-butyl ester

[1-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-4-ylmethyl]-carbamic acid tert-butyl ester

3-(2-Chloro-6-methyl-pyrimidin-4-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

4-(2-Chloro-6-methyl-pyrimidin-4-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

3-[(2-Chloro-6-methyl-pyrimidin-4-yl)-methyl-amino]-piperidine-1-carboxylic acid tert-butyl ester

4-[(2-Chloro-6-methyl-pyrimidin-4-yl)-methyl-amino]-piperidine-1-carboxylic acid tert-butyl ester

2-[(2-Chloro-6-methyl-pyrimidin-4-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

3-[(2-Chloro-6-methyl-pyrimidin-4-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

4-[(2-Chloro-6-methyl-pyrimidin-4-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

(R)-3-(2-Methylsulfanyl-pyrimidin-4-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(2-Methylsulfanyl-pyrimidin-4-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-[(2-Methylsulfanyl-pyrimidin-4-ylamino)-methyl]-pyrrolidine-1-carboxylic acid tert-butyl ester

(R)-3-(2-Methylsulfanyl-pyrimidin-4-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(2-Methylsulfanyl-pyrimidin-4-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-Methylsulfanyl-4-(pyrrolidin-2-ylmethoxy)-pyrimidine hydrochloride

1-(2-Methylsulfanyl-pyrimidin-4-yl)-pyrrolidin-3-ol

(R)-1-(2-Methylsulfanyl-pyrimidin-4-yl)-pyrrolidin-3-ol

(S)-1-(2-Methylsulfanyl-pyrimidin-4-yl)-pyrrolidin-3-ol

4-(2-Methylsulfanyl-pyrimidin-4-yl)-piperazine-1-carboxylic acid tert-butyl ester

3-Methyl-4-(2-methylsulfanyl-pyrimidin-4-yl)-piperazine-1-carboxylic acid tert-butyl ester

4-(2-Methyl-piperazin-1-yl)-2-methylsulfanyl-pyrimidine hydrochloride

2-Methyl-4-(2-methylsulfanyl-pyrimidin-4-yl)-piperazine-1-carboxylic acid tert-butyl ester

4-(3-Methyl-piperazin-1-yl)-2-methylsulfanyl-pyrimidine hydrochloride

4-(2-Methylsulfanyl-pyrimidin-4-yl)-piperazine-1,3-dicarboxylic acid 1-tert-butyl ester

1-(2-Methylsulfanyl-pyrimidin-4-yl)-piperidine-3-carboxylic acid

1-(2-Methylsulfanyl-pyrimidin-4-yl)-piperidine-4-carboxylic acid

1-(2-Methylsulfanyl-pyrimidin-4-yl)-piperidin-3-ol

1-(2-Methylsulfanyl-pyrimidin-4-yl)-piperidin-4-ol

[1-(2-Methylsulfanyl-pyrimidin-4-yl)-piperidin-2-yl]-methanol

[1-(2-Methylsulfanyl-pyrimidin-4-yl)-piperidin-3-yl]-methanol

[1-(2-Methylsulfanyl-pyrimidin-4-yl)-piperidin-4-yl]-methanol

[1-(2-Methylsulfanyl-pyrimidin-4-yl)-piperidin-3-yl]-carbamic acid tert-butyl ester

1-(2-Methylsulfanyl-pyrimidin-4-yl)-piperidin-3-ylamine hydrochloride

[1-(2-Methylsulfanyl-pyrimidin-4-yl)-piperidin-4-yl]-carbamic acid tert-butyl ester

1-(2-Methylsulfanyl-pyrimidin-4-yl)-piperidin-4-ylamine hydrochloride

Methyl-[1-(2-methylsulfanyl-pyrimidin-4-yl)-piperidin-4-yl]-carbamic acid tert-butyl ester

Methyl-[1-(2-methylsulfanyl-pyrimidin-4-yl)-piperidin-4-yl]-amine hydrochloride

C-[1-(2-Methylsulfanyl-pyrimidin-4-yl)-piperidin-3-yl]-methylamine hydrochloride

C-[1-(2-Methylsulfanyl-pyrimidin-4-yl)-piperidin-2-yl]-methylamine hydrochloride

[1-(2-Methylsulfanyl-pyrimidin-4-yl)-piperidin-4-ylmethyl]-carbamic acid tert-butyl ester

3-(2-Methylsulfanyl-pyrimidin-4-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

4-(2-Methylsulfanyl-pyrimidin-4-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

2-[(2-Methylsulfanyl-pyrimidin-4-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

3-[(2-Methylsulfanyl-pyrimidin-4-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

4-[(2-Methylsulfanyl-pyrimidin-4-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

3-[Methyl-(2-methylsulfanyl-pyrimidin-4-yl)-amino]-piperidine-1-carboxylic acid tert-butyl ester

4-[Methyl-(2-methylsulfanyl-pyrimidin-4-yl)-amino]-piperidine-1-carboxylic acid tert-butyl ester

3-(2-Methylsulfanyl-pyrimidin-4-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

4-(2-Methylsulfanyl-pyrimidin-4-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

2-Methylsulfanyl-4-(piperidin-2-ylmethoxy)-pyrimidine hydrochloride

4-(2-Methylsulfanyl-pyrimidin-4-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(6-Chloro-2-methylsulfanyl-pyrimidin-4-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-pyrrolidin-3-yl-amine hydrochloride

(R)-3-(6-Chloro-2-methylsulfanyl-pyrimidin-4-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(6-Chloro-2-methylsulfanyl-pyrimidin-4-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-[(6-Chloro-2-methylsulfanyl-pyrimidin-4-ylamino)-methyl]-pyrrolidine-1-carboxylic acid tert-butyl ester

1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-pyrrolidin-3-ol

(R)-1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-pyrrolidin-3-ol

(S)-1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-pyrrolidin-3-ol

4-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperazine-1-carboxylic acid tert-butyl ester

4-Chloro-2-methylsulfanyl-6-piperazin-1-yl-pyrimidine hydrochloride

4-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-3-methyl-piperazine-1-carboxylic acid tert-butyl ester

4-Chloro-6-(2-methyl-piperazin-1-yl)-2-methylsulfanyl-pyrimidine hydrochloride

4-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-2-methyl-piperazine-1-carboxylic acid tert-butyl ester

4-Chloro-6-(3-methyl-piperazin-1-yl)-2-methylsulfanyl-pyrimidine hydrochloride

4-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperazine-1,3-dicarboxylic acid 1-tert-butyl ester

1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidine-2-carboxylic acid

1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidine-4-carboxylic acid

1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidin-3-ol

1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidin-4-ol

[1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidin-2-yl]-methanol

[1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidin-3-yl]-methanol

[1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidin-4-yl]-methanol

[1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidin-3-yl]-carbamic acid tert-butyl ester

1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidin-3-ylamine hydrochloride

[1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidin-4-yl]-carbamic acid tert-butyl ester

1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidin-4-ylamine hydrochloride

[1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidin-4-yl]-methyl-carbamic acid tert-butyl ester

[1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidin-4-yl]-methyl-amine hydrochloride

[1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidin-3-ylmethyl]-carbamic acid tert-butyl ester

[1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidin-2-ylmethyl]-carbamic acid tert-butyl ester

[1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidin-3-yl]-methyl-carbamic acid tert-butyl ester

[1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidin-3-yl]-methyl-amine hydrochloride

3-(6-Chloro-2-methylsulfanyl-pyrimidin-4-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

4-(6-Chloro-2-methylsulfanyl-pyrimidin-4-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

2-[(6-Chloro-2-methylsulfanyl-pyrimidin-4-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

3-[(6-Chloro-2-methylsulfanyl-pyrimidin-4-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

4-[(6-Chloro-2-methylsulfanyl-pyrimidin-4-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

3-[(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-methyl-amino]-piperidine-1-carboxylic acid tert-butyl ester

4-[(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-methyl-amino]-piperidine-1-carboxylic acid tert-butyl ester

3-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

4-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

3-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

4-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

(R)-3-(4,6-Dimethyl-pyrimidin-2-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-(4,6-Dimethyl-pyrimidin-2-yloxymethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

1-(4,6-Dimethyl-pyrimidin-2-yl)-pyrrolidin-3-ol

(R)-1-(4,6-Dimethyl-pyrimidin-2-yl)-pyrrolidin-3-ol

(S)-1-(4,6-Dimethyl-pyrimidin-2-yl)-pyrrolidin-3-ol

2-[(4,6-Dimethyl-pyrimidin-2-ylamino)-methyl]-pyrrolidine-1-carboxylic acid tert-butyl ester

[1-(4,6-Dimethyl-pyrimidin-2-yl)-piperidin-3-yl]-methyl-carbamic acid tert-butyl ester

3-[(4,6-Dimethyl-pyrimidin-2-yl)-methyl-amino]-piperidine-1-carboxylic acid tert-butyl ester

(S)-3-(5-Fluoro-pyrimidin-2-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

(R)-3-(5-Fluoro-pyrimidin-2-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(5-Fluoro-pyrimidin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

(5-Fluoro-pyrimidin-2-yl)-(S)-pyrrolidin-3-yl-amine hydrochloride

(R)-3-(5-Fluoro-pyrimidin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

1-(5-Fluoro-pyrimidin-2-yl)-pyrrolidin-3-ol

(R)-1-(5-Fluoro-pyrimidin-2-yl)-pyrrolidin-3-ol

(S)-1-(5-Fluoro-pyrimidin-2-yl)-pyrrolidin-3-ol

2-[(5-Fluoro-pyrimidin-2-ylamino)-methyl]-pyrrolidine-1-carboxylic acid tert-butyl ester

5-Fluoro-2-(pyrrolidin-2-ylmethoxy)-pyrimidine hydrochloride

[1-(5-Fluoro-pyrimidin-2-yl)-piperidin-4-yl]-methyl-amine hydrochloride

[1-(5-Fluoro-pyrimidin-2-yl)-piperidin-3-yl]-methyl-amine hydrochloride

4-[(5-Fluoro-pyrimidin-2-yl)-methyl-amino]-piperidine-1-carboxylic acid tert-butyl ester

3-[(5-Fluoro-pyrimidin-2-yl)-methyl-amino]-piperidine-1-carboxylic acid tert-butyl ester

[1-(5-Fluoro-pyrimidin-2-yl)-piperidin-3-ylmethyl]-carbamic acid tert-butyl ester

[1-(5-Fluoro-pyrimidin-2-yl)-piperidin-4-ylmethyl]-carbamic acid tert-butyl ester

2-[(5-Fluoro-pyrimidin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

3-[(5-Fluoro-pyrimidin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

[1-(5-Fluoro-pyrimidin-2-yl)-piperidin-3-yl]-carbamic acid tert-butyl ester

5-Fluoro-2-(2-methyl-piperazin-1-yl)-pyrimidine hydrochloride

5-Fluoro-2-(3-methyl-piperazin-1-yl)-pyrimidine hydrochloride

(S)-3-(5-Chloro-pyrimidin-2-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

(R)-3-(5-Chloro-pyrimidin-2-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(5-Chloro-pyrimidin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(5-Chloro-pyrimidin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

(R)-3-(5-Chloro-pyrimidin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

1-(5-Chloro-pyrimidin-2-yl)-pyrrolidin-3-ol

(R)-1-(5-Chloro-pyrimidin-2-yl)-pyrrolidin-3-ol

(S)-1-(5-Chloro-pyrimidin-2-yl)-pyrrolidin-3-ol

2-(5-Chloro-pyrimidin-2-yloxymethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

[1-(5-Chloro-pyrimidin-2-yl)-piperidin-4-yl]-methyl-amine hydrochloride

[1-(5-Chloro-pyrimidin-2-yl)-piperidin-3-yl]-methyl-amine hydrochloride

4-[(5-Chloro-pyrimidin-2-yl)-methyl-amino]-piperidine-1-carboxylic acid tert-butyl ester

3-[(5-Chloro-pyrimidin-2-yl)-methyl-amino]-piperidine-1-carboxylic acid tert-butyl ester

C-[1-(5-Chloro-pyrimidin-2-yl)-piperidin-2-yl]-methylamine hydrochloride

[1-(5-Chloro-pyrimidin-2-yl)-piperidin-4-ylmethyl]-carbamic acid tert-butyl ester

2-[(5-Chloro-pyrimidin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

3-[(5-Chloro-pyrimidin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

2-Chloro-4,6-dimethyl-pyrimidine

4-[(5-Chloro-pyrimidin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

4-(5-Chloro-pyrimidin-2-yl)-3-methyl-piperazine-1-carboxylic acid tert-butyl ester

4-(5-Chloro-pyrimidin-2-yl)-2-methyl-piperazine-1-carboxylic acid tert-butyl ester

4-Chloro-2-methylsulfanyl-pyrimidine

[1-(5-Chloro-pyrimidin-2-yl)-piperidin-3-yl]-carbamic acid tert-butyl ester

(1r,4r)-4-(6-chloropyrimidin-4-ylamino)cyclohexanol

2,4-Dichloro-6-methyl-pyrimidine

(1r,4r)-4-(pyrimidin-2-ylamino)cyclohexanol

(1r,4r)-4-(5-chloropyrimidin-2-ylamino)cyclohexanol

2,4-Dichloro-5-methyl-pyrimidine

4,6-Dichloro-2-methylsulfanyl-pyrimidine

(1r,4r)-4-(4,6-dimethylpyrimidin-2-ylamino)cyclohexanol

(1r,4r)-4-(5-fluoropyrimidin-2-ylamino)cyclohexanol

2-Chloro-benzothiazole

(1r,4r)-4-(4-methylpyrimidin-2-ylamino)cyclohexanol

(1r,4r)-4-(4-chloro-5-methylpyrimidin-2-ylamino)cyclohexanol

3-Methyl-thiophene-2-sulfonic acid

(1r,4r)-4-(4-chloro-6-methylpyrimidin-2-ylamino)cyclohexanol

(1r,4r)-4-(6-chloro-2-(methylthio)pyrimidin-4-ylamino)cyclohexanol

5-Bromo-thiophene-2-sulfonyl chloride

(1r,4r)-4-(4-chloropyrimidin-2-ylamino)cyclohexanol

2-[(6-Chloro-pyrimidin-4-ylamino)-methyl]-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(6-Chloro-pyrimidin-4-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

(R)-3-(6-Chloro-pyrimidin-4-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

4-Chloro-6-((R)-pyrrolidin-3-yloxy)-pyrimidine hydrochloride

(S)-1-(6-Chloro-pyrimidin-4-yl)-pyrrolidin-3-ol

2-Bromo-1-thiophen-2-yl-ethanone

2-Bromo-1-(1H-pyrrol-2-yl)-ethanone

(R)-1-(6-Chloro-pyrimidin-4-yl)-pyrrolidin-3-ol

4-(6-Chloro-pyrimidin-4-yl)-3-methyl-piperazine-1-carboxylic acid tert-butyl ester

[1-(6-Chloro-pyrimidin-4-yl)-piperidin-4-yl]-methyl-carbamic acid tert-butyl ester

[1-(6-Chloro-pyrimidin-4-yl)-piperidin-4-yl]-methyl-amine hydrochloride

2-Methoxy-3-methyl-pyrazine

[1-(6-Chloro-pyrimidin-4-yl)-piperidin-3-yl]-methyl-carbamic acid tert-butyl ester

4-[(6-Chloro-pyrimidin-4-yl)-methyl-amino]-piperidine-1-carboxylic acid tert-butyl ester

3-[(6-Chloro-pyrimidin-4-yl)-methyl-amino]-piperidine-1-carboxylic acid tert-butyl ester

(6-Chloro-pyrimidin-4-yl)-methyl-piperidin-3-yl-amine hydrochloride

1-(6-Chloro-pyrimidin-4-yl)-piperidine-2-carboxylic acid

1-(6-Chloro-pyrimidin-4-yl)-piperidine-3-carboxylic acid

2-(Pyrimidin-2-ylaminomethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(Pyrimidin-2-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

(R)-3-(Pyrimidin-2-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

1-Pyrimidin-2-yl-pyrrolidin-3-ol

3-(Methyl-pyrimidin-2-yl-amino)-piperidine-1-carboxylic acid tert-butyl ester

Methyl-(1-pyrimidin-2-yl-piperidin-3-yl)-carbamic acid tert-butyl ester

2-[(4-Chloro-pyrimidin-2-ylamino)-methyl]-pyrrolidine-1-carboxylic acid tert-butyl ester

[1-(4-Chloro-pyrimidin-2-yl)-piperidin-4-yl]-methyl-carbamic acid tert-butyl ester

[1-(4-Chloro-pyrimidin-2-yl)-piperidin-3-yl]-methyl-carbamic acid tert-butyl ester

3-[(4-Chloro-pyrimidin-2-yl)-methyl-amino]-piperidine-1-carboxylic acid tert-butyl ester

[1-(4-Chloro-pyrimidin-2-yl)-piperidin-2-yl]-methanol

(R)-3-(2-Chloro-pyrimidin-4-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(2-Chloro-pyrimidin-4-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

(R)-1-(2-Chloro-pyrimidin-4-yl)-pyrrolidin-3-ol

(S)-1-(2-Chloro-pyrimidin-4-yl)-pyrrolidin-3-ol

4-(2-Chloro-pyrimidin-4-yl)-3-methyl-piperazine-1-carboxylic acid tert-butyl ester

2-Chloro-4-(2-methyl-piperazin-1-yl)-pyrimidine hydrochloride

4-(2-Chloro-pyrimidin-4-yl)-2-methyl-piperazine-1-carboxylic acid tert-butyl ester

4-(2-Chloro-pyrimidin-4-yl)-piperazine-1,3-dicarboxylic acid 1-tert-butyl ester

3-Bromomethyl-6-chloro-pyridazine

1-(2-Chloro-pyrimidin-4-yl)-piperidine-2-carboxylic acid

1-(2-Chloro-pyrimidin-4-yl)-piperidine-3-carboxylic acid

2-Bromo-4-bromomethyl-pyridine

[1-(2-Chloro-pyrimidin-4-yl)-piperidin-4-yl]-methanol

[1-(2-Chloro-pyrimidin-4-yl)-piperidin-3-yl]-methyl-carbamic acid tert-butyl ester

[1-(2-Chloro-pyrimidin-4-yl)-piperidin-4-yl]-methyl-carbamic acid tert-butyl ester

[1-(2-Chloro-pyrimidin-4-yl)-piperidin-4-yl]-methyl-amine hydrochloride

3-[(2-Chloro-pyrimidin-4-yl)-methyl-amino]-piperidine-1-carboxylic acid tert-butyl ester

4-Bromomethyl-2-chloro-pyrimidine

4-[(2-Chloro-pyrimidin-4-yl)-methyl-amino]-piperidine-1-carboxylic acid tert-butyl ester

(2-Chloro-pyrimidin-4-yl)-methyl-piperidin-4-yl-amine hydrochloride

4-(2-Chloro-pyrimidin-4-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-(methylthio)-4,6-bis(N-tert-butyloxy-carbonyl-piperidin-4-yloxy)pyrimidine

2-Methylsulfanyl-4,6-bis-(piperidin-3-yloxy)-pyrimidine dihydrochloride

2-Methylsulfanyl-4,6-bis-(piperidin-2-yloxy)-pyrimidine dihydrochloride

N,N -Bis-(6-chloro-pyrimidin-4-yl)-cyclohexane-1,4-diamine

tert-butyl-4-((2-((1-(tert-butoxycarbonyl)piperidin-4-yl)methoxy)pyrimidin-4-yloxy)methyl)piperidine-1-carboxylate

tert-butyl-2-((2-((1-(tert-butoxycarbonyl)pyrrolidin-2-yl)methoxy)pyrimidin-4-yloxy)methyl)pyrrolidine-1-carboxylate

5-Chloro-2-(piperidin-2-ylmethoxy)-pyrimidine hydrochloride

5-Chloro-2-(piperidin-3-ylmethoxy)-pyrimidine hydrochloride

5-Chloro-2-(piperidin-4-ylmethoxy)-pyrimidine hydrochloride

3-(5-Chloro-pyrimidin-2-yloxy)-piperidine-1-carboxylic acid tert-butylester

2-Chloro-3H-imidazo[4,5-b]pyridine

2-Bromo-pyridin-3-ol N-oxide

2-Chloro-5-methoxymethyl-pyridine

5-Chloro-2-(piperidin-3-yloxy)-pyrimidine hydrochloride

2-Chloro-5-ethoxymethyl-pyridine

5-Chloro-2-(piperidin-4-yloxy)-pyrimidine hydrochloride

4-(5-Chloro-pyrimidin-2-yl)-piperazine-2-carboxylic acid

1-(5-Chloro-pyrimidin-2-yl)-piperazine-2-carboxylic acid hydrochloride

1-(5-Chloro-pyrimidin-2-yl)-piperidin-4-ylamine hydrochloride

4-(5-Chloro-pyrimidin-2-yl)-[1,4]diazepane-1-carboxylic acid tert-butyl ester

1-(5-Chloro-pyrimidin-2-yl)-[1,4]diazepane hydrochloride

4,6-Dimethyl-2-(piperidin-2-ylmethoxy)-pyrimidine hydrochloride

4,6-Dimethyl-2-(piperidin-3-ylmethoxy)-pyrimidine hydrochloride

(6-Chloro-pyridazin-3-ylmethyl)-isopropyl-amine

4-(4,6-Dimethyl-pyrimidin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

4,6-Dimethyl-2-(piperidin-4-ylmethoxy)-pyrimidine hydrochloride

4,6-Dimethyl-2-(piperidin-3-yloxy)-pyrimidine hydrochloride

4,6-Dimethyl-2-(piperidin-4-yloxy)-pyrimidine hydrochloride

4-(4,6-Dimethyl-pyrimidin-2-yl)-piperazine-2-carboxylic acid

(6-Bromo-pyridin-3-ylmethyl)-cyclopropyl-amine

1-(4,6-Dimethyl-pyrimidin-2-yl)-piperazine-2-carboxylic acid hydrochloride

5-Fluoro-2-(piperidin-2-ylmethoxy)-pyrimidine hydrochloride

5-Fluoro-2-(piperidin-3-ylmethoxy)-pyrimidine hydrochloride

5-Fluoro-2-(piperidin-4-ylmethoxy)-pyrimidine hydrochloride

5-Fluoro-2-(piperidin-3-yloxy)-pyrimidine hydrochloride

5-Fluoro-2-(piperidin-4-yloxy)-pyrimidine hydrochloride

4-(5-Fluoro-pyrimidin-2-yl)-piperazine-2-carboxylic acid

1-(5-Fluoro-pyrimidin-2-yl)-piperazine-2-carboxylic acid hydrochloride

[1-(5-Fluoro-pyrimidin-2-yl)-piperidin-2-yl]-methanol

3-(5-Fluoro-pyrimidin-2-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

1-(5-Fluoro-pyrimidin-2-yl)-piperidin-4-ylamine hydrochloride

4-(5-Fluoro-pyrimidin-2-yl)-[1,4]diazepane-1-carboxylic acid tert-butyl ester

1-(5-Fluoro-pyrimidin-2-yl)-[1,4]diazepane hydrochloride

2-(Piperidin-2-ylmethoxy)-pyrimidine hydrochloride

4-Pyrimidin-2-yl-piperazine-2-carboxylic acid

1-Pyrimidin-2-yl-piperazine-2-carboxylic acid hydrochloride

(4-Methyl-pyrimidin-2-yl)-pyrrolidin-3-yl-amine hydrochloride

(4-Methyl-pyrimidin-2-yl)-(R)-pyrrolidin-3-yl-amine hydrochloride

(4-Methyl-pyrimidin-2-yl)-(S)-pyrrolidin-3-yl-amine hydrochloride

(4-Methyl-pyrimidin-2-yl)-pyrrolidin-2-ylmethyl-amine hydrochloride

4-Methyl-2-((R)-pyrrolidin-3-yloxy)-pyrimidine hydrochloride

(2-Bromo-pyridin-4-ylmethyl)-ethyl-amine

4-Methyl-2-((S)-pyrrolidin-3-yloxy)-pyrimidine hydrochloride

4-Methyl-2-(pyrrolidin-2-ylmethoxy)-pyrimidine hydrochloride

1-(4-Methyl-pyrimidin-2-yl)-azetidine-3-carboxylic acid

4-(4-Methyl-pyrimidin-2-yl)-[1,4]diazepane-1-carboxylic acid tert-butyl ester

1-(4-Methyl-pyrimidin-2-yl)-[1,4]diazepane hydrochloride

3-Methyl-4-(4-methyl-pyrimidin-2-yl)-piperazine-1-carboxylic acid tert-butyl ester

4-Methyl-2-(2-methyl-piperazin-1-yl)-pyrimidine hydrochloride

4-Methyl-2-(3-methyl-piperazin-1-yl)-pyrimidine hydrochloride

4-(4-Methyl-pyrimidin-2-yl)-piperazine-1,3-dicarboxylic acid 1-tert-butyl ester

1-(4-Methyl-pyrimidin-2-yl)-piperazine-2-carboxylic acid hydrochloride

4-(4-Methyl-pyrimidin-2-yl)-piperazine-2-carboxylic acid

1-(4-Methyl-pyrimidin-2-yl)-piperidine-2-carboxylic acid

1-(4-Methyl-pyrimidin-2-yl)-piperidin-3-ylamine hydrochloride

1-(4-Methyl-pyrimidin-2-yl)-piperidin-4-ylamine hydrochloride

Methyl-[1-(4-methyl-pyrimidin-2-yl)-piperidin-4-yl]-amine hydrochloride

[1-(4-Methyl-pyrimidin-2-yl)-piperidin-3-ylmethyl]-carbamic acid tert-butyl ester

C-[1-(4-Methyl-pyrimidin-2-yl)-piperidin-3-yl]-methylamine hydrochloride

[1-(4-Methyl-pyrimidin-2-yl)-piperidin-2-ylmethyl]-carbamic acid tert-butyl ester

C-[1-(4-Methyl-pyrimidin-2-yl)-piperidin-2-yl]-methylamine hydrochloride

C-[1-(4-Methyl-pyrimidin-2-yl)-piperidin-4-yl]-methylamine hydrochloride

Methyl-[1-(4-methyl-pyrimidin-2-yl)-piperidin-3-yl]-amine hydrochloride

(4-Methyl-pyrimidin-2-yl)-piperidin-3-yl-amine hydrochloride

(4-Methyl-pyrimidin-2-yl)-piperidin-4-yl-amine hydrochloride

(4-Methyl-pyrimidin-2-yl)-piperidin-2-ylmethyl-amine hydrochloride

(4-Methyl-pyrimidin-2-yl)-piperidin-3-ylmethyl-amine hydrochloride

(4-Methyl-pyrimidin-2-yl)-piperidin-4-ylmethyl-amine hydrochloride

Methyl-(4-methyl-pyrimidin-2-yl)-piperidin-3-yl-amine hydrochloride

Methyl-(4-methyl-pyrimidin-2-yl)-piperidin-4-yl-amine hydrochloride

4-Methyl-2-(piperidin-3-yloxy)-pyrimidine hydrochloride

4-Methyl-2-(piperidin-4-yloxy)-pyrimidine hydrochloride

4-Methyl-2-(piperidin-2-ylmethoxy)-pyrimidine hydrochloride

4-Methyl-2-(piperidin-3-ylmethoxy)-pyrimidine hydrochloride

4-Methyl-2-(piperidin-4-ylmethoxy)-pyrimidine hydrochloride

(4-Chloro-5-methyl-pyrimidin-2-yl)-pyrrolidin-3-yl-amine hydrochloride

(4-Chloro-5-methyl-pyrimidin-2-yl)-(R)-pyrrolidin-3-yl-amine hydrochloride

(4-Chloro-5-methyl-pyrimidin-2-yl)-(S)-pyrrolidin-3-yl-amine hydrochloride

(4-Chloro-5-methyl-pyrimidin-2-yl)-pyrrolidin-2-ylmethyl-amine hydrochloride

4-Chloro-5-methyl-2-((R)-pyrrolidin-3-yloxy)-pyrimidine hydrochloride

4-Chloro-5-methyl-2-((S)-pyrrolidin-3-yloxy)-pyrimidine hydrochloride

2-(4-Chloro-5-methyl-pyrimidin-2-yloxymethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

4-Chloro-5-methyl-2-(pyrrolidin-2-ylmethoxy)-pyrimidine hydrochloride

1-(4-Chloro-5-methyl-pyrimidin-2-yl)-azetidine-3-carboxylic acid

4-(4-Chloro-5-methyl-pyrimidin-2-yl)-[1,4]diazepane-1-carboxylic acid tert-butyl ester

1-(4-Chloro-5-methyl-pyrimidin-2-yl)-[1,4]diazepane hydrochloride

1-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperazine-2-carboxylic acid hydrochloride

4-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperazine-2-carboxylic acid

1-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidin-4-ylamine hydrochloride

C-[1-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidin-3-yl]-methylamine hydrochloride

C-[1-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidin-2-yl]-methylamine hydrochloride

[1-(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidin-3-yl]-methyl-carbamic acid tert-butyl ester

(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidin-3-yl-amine hydrochloride

(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidin-4-yl-amine hydrchloride

(4-Chloro-5-methyl-pyrimidin-2-yl)-piperidin-2-ylmethyl-amine hydrochloride

(4-Chloro-5-methyl-pyrimidin-2-yl)-methyl-piperidin-3-yl-amine hydrochloride

(4-Chloro-5-methyl-pyrimidin-2-yl)-methyl-piperidin-4-yl-amine hydrochloride

4-Chloro-5-methyl-2-(piperidin-3-yloxy)-pyrimidine hydrochloride

4-Chloro-5-methyl-2-(piperidin-4-yloxy)-pyrimidine hydrochloride

2-(4-Chloro-5-methyl-pyrimidin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

4-Chloro-5-methyl-2-(piperidin-2-ylmethoxy)-pyrimidine hydrochloride

3-(4-Chloro-5-methyl-pyrimidin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

4-Chloro-5-methyl-2-(piperidin-3-ylmethoxy)-pyrimidine hydrochloride

4-Chloro-5-methyl-2-(piperidin-4-ylmethoxy)-pyrimidine hydrochloride

(4-Chloro-6-methyl-pyrimidin-2-yl)-pyrrolidin-3-yl-amine hydrochloride

(R)-3-(4-Chloro-6-methyl-pyrimidin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

1-Thiazol-2-yl-piperidin-4-ylamine hydrochloride

(4-Chloro-6-methyl-pyrimidin-2-yl)-(R)-pyrrolidin-3-yl-amine hydrochloride

4-(2-Chloro-thiazol-5-ylmethoxy)-piperidine-1-carboxylic acid tert-butyl ester

(4-Chloro-6-methyl-pyrimidin-2-yl)-(S)-pyrrolidin-3-yl-amine hydrochloride

2-[(4-Chloro-6-methyl-pyrimidin-2-ylamino)-methyl]-pyrrolidine-1-carboxylic acid tert-butyl ester

(4-Chloro-6-methyl-pyrimidin-2-yl)-pyrrolidin-2-ylmethyl-amine hydrochloride

3-(2-Chloro-thiazol-5-ylmethoxy)-piperidine dihydrochloride

(R)-3-(4-Chloro-6-methyl-pyrimidin-2-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

4-Chloro-6-methyl-2-((R)-pyrrolidin-3-yloxy)-pyrimidine hydrochloride

3-(2-Chloro-thiazol-5-ylmethoxy)-piperidine-1-carboxylic acid tert-butyl ester

(S)-3-(4-Chloro-6-methyl-pyrimidin-2-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

4-Chloro-6-methyl-2-((S)-pyrrolidin-3-yloxy)-pyrimidine hydrochloride

2-(4-Chloro-6-methyl-pyrimidin-2-yloxymethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

1-(2-Chloro-thiazol-5-ylmethyl)-piperidin-4-ylamine dihydrochloride

4-Chloro-6-methyl-2-(pyrrolidin-2-ylmethoxy)-pyrimidine hydrochloride

(S)-1-(4-Chloro-6-methyl-pyrimidin-2-yl)-pyrrolidin-3-ol

[1-(2-Chloro-thiazol-5-ylmethyl)-piperidin-4-yl]-carbamic acid tert-butyl ester

1-(2-Chloro-thiazol-5-ylmethyl)-piperidin-3-ylamine dihydrochloride

1-(4-Chloro-6-methyl-pyrimidin-2-yl)-azetidine-3-carboxylic acid

4-(4-Chloro-6-methyl-pyrimidin-2-yl)-[1,4]diazepane-1-carboxylic acid tert-butyl ester

[1-(2-Chloro-thiazol-5-ylmethyl)-piperidin-3-yl]-carbamic acid tert-butyl ester

1-(4-Chloro-6-methyl-pyrimidin-2-yl)-[1,4]diazepane hydrochloride

4-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperazine-1-carboxylic acid tert-butyl ester

1-(2-Chloro-thiazol-5-ylmethyl)-piperazine dihydrochloride

4-Chloro-6-methyl-2-piperazin-1-yl-pyrimidine hydrochloride

4-(2-Chloro-thiazol-5-ylmethyl)-piperazine-1-carboxylic acid tert-butyl ester

4-(4-Chloro-6-methyl-pyrimidin-2-yl)-3-methyl-piperazine-1-carboxylic acid tert-butyl ester

4-Chloro-6-methyl-2-(2-methyl-piperazin-1-yl)-pyrimidine hydrochloride

4-(4-Chloro-6-methyl-pyrimidin-2-yl)-2-methyl-piperazine-1-carboxylic acid tert-butyl ester

4-Chloro-6-methyl-2-(3-methyl-piperazin-1-yl)-pyrimidine hydrochloride

4-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperazine-1,3-dicarboxylic acid 1-tert-butyl ester

1-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperazine-2-carboxylic acid hydrochloride

4-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperazine-2-carboxylic acid

1-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidine-2-carboxylic acid

1-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidine-4-carboxylic acid

1-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidin-4-ol

[1-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidin-3-yl]-carbamic acid tert-butyl ester

1-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidin-3-ylamine hydrochloride

1-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidin-4-ylamine hydrochloride

[1-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidin-4-yl]-methyl-carbamic acid tert-butyl ester

[1-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidin-4-yl]-methyl-amine hydrochloride

[1-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidin-3-ylmethyl]-carbamic acid tert-butyl ester

C-[1-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidin-3-yl]-methylamine hydrochloride

[1-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidin-2-ylmethyl]-carbamic acid tert-butyl ester

C-[1-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidin-2-yl]-methylamine hydrochloride

C-[1-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidin-4-yl]-methylamine hydrochloride

[1-(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidin-3-yl]-methyl-amine hydrochloride

3-(4-Chloro-6-methyl-pyrimidin-2-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidin-3-yl-amine hydrochloride

4-(4-Chloro-6-methyl-pyrimidin-2-ylamino)-piperidine-1-carboxylic acid tert-butyl ester

4-(4-Bromo-benzenesulfonylmethyl)-piperidine

(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidin-4-yl-amine hydrochloride

2-[(4-Chloro-6-methyl-pyrimidin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidin-2-ylmethyl-amine hydrochloride

3-(4-Bromo-benzenesulfonylmethyl)-piperidine

3-[(4-Chloro-6-methyl-pyrimidin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidin-3-ylmethyl-amine hydrochloride

4-[(4-Chloro-6-methyl-pyrimidin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

(4-Chloro-6-methyl-pyrimidin-2-yl)-piperidin-4-ylmethyl-amine hydrochloride

(4-Chloro-6-methyl-pyrimidin-2-yl)-methyl-piperidin-3-yl-amine hydrochloride

4-[(4-Chloro-6-methyl-pyrimidin-2-yl)-methyl-amino]-piperidine-1-carboxylic acid tert-butyl ester

(4-Chloro-6-methyl-pyrimidin-2-yl)-methyl-piperidin-4-yl-amine hydrochloride

2-(4-Bromo-benzenesulfonylmethyl)-piperidine

3-(4-Chloro-6-methyl-pyrimidin-2-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

4-Chloro-6-methyl-2-(piperidin-3-yloxy)-pyrimidine hydrochloride

4-(4-Bromo-benzenesulfonyl)-piperidine-1-carboxylic acid tert-butyl ester

4-(4-Chloro-6-methyl-pyrimidin-2-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

4-Chloro-6-methyl-2-(piperidin-4-yloxy)-pyrimidine hydrochloride

3-(4-Bromo-benzenesulfonyl)-piperidine-1-carboxylic acid tert-butyl ester

4-(4-Chloro-6-methyl-pyrimidin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

4-Chloro-6-methyl-2-(piperidin-2-ylmethoxy)-pyrimidine hydrochloride

4-(4-Bromo-benzenesulfonylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(4-Chloro-6-methyl-pyrimidin-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(4-Bromo-benzenesulfonylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

4-Chloro-6-methyl-2-(piperidin-3-ylmethoxy)-pyrimidine hydrochloride

4-Chloro-6-methyl-2-(piperidin-4-ylmethoxy)-pyrimidine hydrochloride

2-(4-Bromo-benzenesulfonylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(2-Chloro-6-methyl-pyrimidin-4-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

(2-Chloro-6-methyl-pyrimidin-4-yl)-pyrrolidin-3-yl-amine hydrochloride

(S)-3-(3-Fluoro-phenylsulfanyl)-pyrrolidine

(2-Chloro-6-methyl-pyrimidin-4-yl)-(R)-pyrrolidin-3-yl-amine hyrochloride

(2-Chloro-6-methyl-pyrimidin-4-yl)-(S)-pyrrolidin-3-yl-amine hydrochloride

(R)-3-(3-Fluoro-phenylsulfanyl)-pyrrolidine

(2-Chloro-6-methyl-pyrimidin-4-yl)-pyrrolidin-2-ylmethyl-amine hydrochloride

3-(3-Fluoro-phenylsulfanyl)-pyrrolidine

(R)-3-(2-Chloro-6-methyl-pyrimidin-4-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-Chloro-4-methyl-6-((R)-pyrrolidin-3-yloxy)-pyrimidine hydrochloride

3-(3-Fluoro-phenylsulfanylmethyl)-pyrrolidine

(S)-3-(2-Chloro-6-methyl-pyrimidin-4-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-Chloro-4-methyl-6-((S)-pyrrolidin-3-yloxy)-pyrimidine hydrochloride

2-(3-Fluoro-phenylsulfanylmethyl)-pyrrolidine

2-(2-Chloro-6-methyl-pyrimidin-4-yloxymethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-(3-Fluoro-phenylsulfanyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-Chloro-4-methyl-6-(pyrrolidin-2-ylmethoxy)-pyrimidine hydrochloride

1-(2-Chloro-6-methyl-pyrimidin-4-yl)-azetidine-3-carboxylic acid

(R)-3-(3-Fluoro-phenylsulfanyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

4-(2-Chloro-6-methyl-pyrimidin-4-yl)-[1,4]diazepane-1-carboxylic acid tert-butyl ester

3-(3-Fluoro-phenylsulfanyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

1-(2-Chloro-6-methyl-pyrimidin-4-yl)-[1,4]diazepane hydrochloride

4-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperazine-2-carboxylic acid

2-Chloro-4-methyl-6-piperazin-1-yl-pyrimidine hydrochloride

3-(3-Fluoro-phenylsulfanylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-Chloro-4-methyl-6-(2-methyl-piperazin-1-yl)-pyrimidine hydrochloride

2-Chloro-4-methyl-6-(3-methyl-piperazin-1-yl)-pyrimidine hydrochloride

2-(3-Fluoro-phenylsulfanylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

1-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperazine-2-carboxylic acid hydrochloride

4-(3-Fluoro-phenylsulfanyl)-piperidine

1-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidine-2-carboxylic acid

3-(3-Fluoro-phenylsulfanyl)-piperidine

4-(3-Fluoro-phenylsulfanylmethyl)-piperidine

3-(3-Fluoro-phenylsulfanylmethyl)-piperidine

2-(3-Fluoro-phenylsulfanylmethyl)-piperidine

(6-Chloro-2-methanesulfonyl-pyrimidin-4-yl)-ethyl-amine

4-(3-Fluoro-phenylsulfanyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(3-Fluoro-phenylsulfanyl)-piperidine-1-carboxylic acid tert-butyl ester

4-(3-Fluoro-phenylsulfanylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(3-Fluoro-phenylsulfanylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-(3-Fluoro-phenylsulfanylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

(S)-3-(3-Fluoro-benzenesulfinyl)-pyrrolidine

(R)-3-(3-Fluoro-benzenesulfinyl)-pyrrolidine

3-(3-Fluoro-benzenesulfinyl)-pyrrolidine

3-(3-Fluoro-benzenesulfinylmethyl)-pyrrolidine

2-(3-Fluoro-benzenesulfinylmethyl)-pyrrolidine

(S)-3-(3-Fluoro-benzenesulfinyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

(R)-3-(3-Fluoro-benzenesulfinyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(3-Fluoro-benzenesulfinyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(3-Fluoro-benzenesulfinylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

1-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidine-4-carboxylic acid

1-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-3-ol

[1-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-2-yl]-methanol

[1-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-4-yl]-methanol

[1-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-3-yl]-carbamic acid tert-butyl ester

1-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-3-ylamine hydrochloride

1-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-4-ylamine hydrochloride

[1-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-3-yl]-methyl-carbamic acid tert-butyl ester

[1-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-3-yl]-methyl-amine hydrochloride

[1-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-4-yl]-methyl-amine hydrochloride

C-[1-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-2-yl]-methylamine hydrochloride

C-[1-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-3-yl]-methylamine hydrochloride

2-(3-Fluoro-benzenesulfinylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

C-[1-(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-4-yl]-methylamine hydrochloride

4-(3-Fluoro-benzenesulfinyl)-piperidine

(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-3-yl-amine hydrochloride

(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-4-yl-amine hydrochloride

(2-Chloro-6-methyl-pyrimidin-4-yl)-methyl-piperidin-3-yl-amine hydrochloride

3-(3-Fluoro-benzenesulfinyl)-piperidine

(2-Chloro-6-methyl-pyrimidin-4-yl)-methyl-piperidin-4-yl-amine hydrochloride

4-(3-Fluoro-benzenesulfinylmethyl)-piperidine

(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-2-ylmethyl-amine hydrochloride

(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-3-ylmethyl-amine hydrochloride

3-(3-Fluoro-benzenesulfinylmethyl)-piperidine

(2-Chloro-6-methyl-pyrimidin-4-yl)-piperidin-4-ylmethyl-amine hydrochloride

2-(3-Fluoro-benzenesulfinylmethyl)-piperidine

3-(2-Chloro-6-methyl-pyrimidin-4-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

2-Chloro-4-methyl-6-(piperidin-3-yloxy)-pyrimidine hydrochloride

4-(3-Fluoro-benzenesulfinyl)-piperidine-1-carboxylic acid tert-butyl ester

(4-Chloro-6-methyl-pyrimidin-2-yl)-ethyl-a

4-(2-Chloro-6-methyl-pyrimidin-4-yloxy)-piperidine-1-carboxylic acid tert-butyl ester

3-(3-Fluoro-benzenesulfinyl)-piperidine-1-carboxylic acid tert-butyl ester

2-Chloro-4-methyl-6-(piperidin-4-yloxy)-pyrimidine hydrochloride

2-(2-Chloro-6-methyl-pyrimidin-4-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

4-(3-Fluoro-benzenesulfinylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

(4-Chloro-6-methyl-pyrimidin-2-yl)-cyclopropyl-amine

2-Chloro-4-methyl-6-(piperidin-2-ylmethoxy)-pyrimidine hydrochloride

3-(3-Fluoro-benzenesulfinylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(2-Chloro-6-methyl-pyrimidin-4-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-(3-Fluoro-benzenesulfinylmethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-Chloro-4-methyl-6-(piperidin-3-ylmethoxy)-pyrimidine hydrochloride

4-(2-Chloro-6-methyl-pyrimidin-4-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

(S)-3-(3-Fluoro-benzenesulfonyl)-pyrrolidine

2-Chloro-4-methyl-6-(piperidin-4-ylmethoxy)-pyrimidine hydrochloride

(R)-3-(3-Fluoro-benzenesulfonyl)-pyrrolidine

[4-(2-Chloro-6-methyl-pyrimidin-4-ylamino)-cyclohexyl]-carbamic acid tert-butyl ester

3-(3-Fluoro-benzenesulfonyl)-pyrrolidine

N-(2-Chloro-6-methyl-pyrimidin-4-yl)-cyclohexane-1,4-diamine hydrochloride

3-(3-Fluoro-benzenesulfonylmethyl)-pyrrolidine

2-(3-Fluoro-benzenesulfonylmethyl)-pyrrolidine

[2-(2-Chloro-6-methyl-pyrimidin-4-ylamino)-cyclohexyl]-carbamic acid tert-butyl ester

(S)-3-(3-Fluoro-benzenesulfonyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

N-(2-Chloro-6-methyl-pyrimidin-4-yl)-cyclohexane-1,2-diamine hydrochloride

4-(2-Chloro-6-methyl-pyrimidin-4-ylamino)-cyclohexanol

(R)-3-(3-Fluoro-benzenesulfonyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

(2-Methylsulfanyl-pyrimidin-4-yl)-(R)-pyrrolidin-3-yl-amine hydrochloride

3-(3-Fluoro-benzenesulfonyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

(2-Methylsulfanyl-pyrimidin-4-yl)-(S)-pyrrolidin-3-yl-amine hydrochloride

(2-Methylsulfanyl-pyrimidin-4-yl)-pyrrolidin-2-ylmethyl-amine hydrochloride

3-(3-Fluoro-benzenesulfonylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-Methylsulfanyl-4-((R)-pyrrolidin-3-yloxy)-pyrimidine hydrochloride

2-Methylsulfanyl-4-((S)-pyrrolidin-3-yloxy)-pyrimidine hydrochloride

2-(3-Fluoro-benzenesulfonylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-(2-Methylsulfanyl-pyrimidin-4-yloxymethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

4-(3-Fluoro-benzenesulfonyl)-piperidine

1-(2-Methylsulfanyl-pyrimidin-4-yl)-azetidine-3-carboxylic acid

3-(3-Fluoro-benzenesulfonyl)-piperidine

(3-Chloro-quinoxalin-2-yl)-ethyl-amine

(3-Chloro-quinoxalin-2-yl)-isopropyl-amine

Benzo[1,3]dioxole-5-carboxylic acid

piperidin-3-ylmethyl trifluoromethanesulfonate 906073-55-0

piperidin-2-ylmethyl trifluoromethanesulfonate 127075-48-3

tert-butyl 4-(trifluoromethylsulfonyloxy)piperidine-1-carboxylate

tert-butyl 2-((trifluoromethylsulfonyloxy)methyl)piperidine-1-carboxylate

(R)-3-Methylamino-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-Methylamino-pyrrolidine-1-carboxylic acid tert-butyl ester

3-Methylaminomethyl-pyrrolidine-1-carboxylic acid tert-butyl ester

2-Methylaminomethyl-pyrrolidine-1-carboxylic acid isopropyl ester

Methyl-(R)-pyrrolidin-3-yl-amine

Methyl-(S)-pyrrolidin-3-yl-amine

Methyl-piperidin-4-ylmethyl-amine

Methyl-piperidin-3-ylmethyl-amine

Methyl-piperidin-2-ylmethyl-amine

3-Methylamino-piperidine-1-carboxylic acid tert-butyl ester

4-Methylaminomethyl-piperidine-1-carboxylic acid tert-butyl ester

3-Methylaminomethyl-piperidine-1-carboxylic acid isopropyl ester

2-Methylaminomethyl-piperidine-1-carboxylic acid tert-butyl ester

(R)-3-Ethylamino-pyrrolidine-1-carboxylic acid tert-butyl ester

(S)-3-Ethylamino-pyrrolidine-1-carboxylic acid tert-butyl ester

3-Ethylamino-pyrrolidine-1-carboxylic acid tert-butyl ester

Ethyl-pyrrolidin-3-yl-amine

Ethyl-pyrrolidin-3-ylmethyl-amine

Ethyl-piperidin-4-ylmethyl-amine

4-(2-Methylsulfanyl-pyrimidin-4-yl)-[1,4]diazepane-1-carboxylic acid tert-butyl ester

1-(2-Methylsulfanyl-pyrimidin-4-yl)-[1,4]diazepane hydrochloride

2-Methylsulfanyl-4-piperazin-1-yl-pyrimidine hydrochloride

1-(2-Methylsulfanyl-pyrimidin-4-yl)-piperazine-2-carboxylic acid hydrochloride

4-(2-Methylsulfanyl-pyrimidin-4-yl)-piperazine-2-carboxylic acid

1-(2-Methylsulfanyl-pyrimidin-4-yl)-piperidine-2-carboxylic acid

[1-(2-Methylsulfanyl-pyrimidin-4-yl)-piperidin-3-ylmethyl]-carbamic acid tert-butyl ester

[1-(2-Methylsulfanyl-pyrimidin-4-yl)-piperidin-2-ylmethyl]-carbamic acid tert-butyl ester

C-[1-(2-Methylsulfanyl-pyrimidin-4-yl)-piperidin-4-yl]-methylamine hydrochloride

Methyl-[1-(2-methylsulfanyl-pyrimidin-4-yl)-piperidin-3-yl]-carbamic acid tert-butyl ester

Methyl-[1-(2-methylsulfanyl-pyrimidin-4-yl)-piperidin-3-yl]-amine hydrochloride

(2-Methylsulfanyl-pyrimidin-4-yl)-piperidin-3-yl-amine hydrochloride

(2-Methylsulfanyl-pyrimidin-4-yl)-piperidin-4-yl-amine hydrochloride

(2-Methylsulfanyl-pyrimidin-4-yl)-piperidin-2-ylmethyl-amine hydrochloride

(2-Methylsulfanyl-pyrimidin-4-yl)-piperidin-3-ylmethyl-amine hydrochloride

(2-Methylsulfanyl-pyrimidin-4-yl)-piperidin-4-ylmethyl-amine hydrochloride

Methyl-(2-methylsulfanyl-pyrimidin-4-yl)-piperidin-3-yl-amine hydrochloride

Methyl-(2-methylsulfanyl-pyrimidin-4-yl)-piperidin-4-yl-amine hydrochloride

2-Methylsulfanyl-4-(piperidin-3-yloxy)-pyrimidine hydrochloride

2-Methylsulfanyl-4-(piperidin-4-yloxy)-pyrimidine hydrochloride

2-(2-Methylsulfanyl-pyrimidin-4-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

3-(2-Methylsulfanyl-pyrimidin-4-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-Methylsulfanyl-4-(piperidin-3-ylmethoxy)-pyrimidine hydrochloride

2-Methylsulfanyl-4-(piperidin-4-ylmethoxy)-pyrimidine hydrochloride

(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-(R)-pyrrolidin-3-yl-amine hydrochloride

(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-(S)-pyrrolidin-3-yl-amine hydrochloride

(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-pyrrolidin-2-ylmethyl-amine hydrochloride

(R)-3-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

4-Chloro-2-methylsulfanyl-6-((R)-pyrrolidin-3-yloxy)-pyrimidine hydrochloride

(S)-3-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yloxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

4-Chloro-2-methylsulfanyl-6-((S)-pyrrolidin-3-yloxy)-pyrimidine hydrochloride

2-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yloxymethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

4-Chloro-2-methylsulfanyl-6-(pyrrolidin-2-ylmethoxy)-pyrimidine hydrochloride

1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-azetidine-3-carboxylic acid

4-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-[1,4]diazepane-1-carboxylic acid tert-butyl ester

1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-[1,4]diazepane hydrochloride

1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperazine-2-carboxylic acid hydrochloride

4-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperazine-2-carboxylic acid

1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidine-3-carboxylic acid

C-[1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidin-3-yl]-methyl-amine hydrochloride

C-[1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidin-2-yl]-methyl-amine hydrochloride

[1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidin-4-ylmethyl]-carbamic acid tert-butyl ester

C-[1-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidin-4-yl]-methyl-amine hydrochloride

(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidin-3-yl-amine hydrochloride

(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidin-4-yl-amine hydrochloride

1-(2-Chloro-thiazol-5-ylmethyl)-piperidine-4-carboxylic acid

1-(2-Chloro-thiazol-5-ylmethyl)-piperidin-4-ol

1-(2-Chloro-thiazol-5-ylmethyl)-piperidin-3-ol

[1-(2-Chloro-thiazol-5-ylmethyl)-piperidin-3-yl]-methanol

4-Thiazol-2-yl-piperazine-1,3-dicarboxylic acid 1-tert-butyl ester

2-(Thiazol-2-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

2-Methyl-1-thiazol-5-ylmethyl-piperazine hydrochloride

3-Methyl-1-thiazol-5-ylmethyl-piperazine hydrochloride

1-Thiazol-5-ylmethyl-piperidin-4-ol

(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidin-2-ylmethyl-amine hydrochloride

1-Thiazol-5-ylmethyl-piperidin-3-ylamine hydrochloride

(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidin-3-ylmethyl-amine hydrochloride

(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-piperidin-4-ylmethyl-amine hydrochloride

(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-methyl-piperidin-3-yl-amine hydrochloride

1-Thiazol-5-ylmethyl-piperidin-4-ylamine hydrochloride

(6-Chloro-2-methylsulfanyl-pyrimidin-4-yl)-methyl-piperidin-4-yl-amine hydrochloride

Methyl-(1-thiazol-5-ylmethyl-piperidin-4-yl)-amine hydrochloride

4-Chloro-2-methylsulfanyl-6-(piperidin-3-yloxy)-pyrimidine hydrochloride

Methyl-(1-thiazol-5-ylmethyl-piperidin-3-yl)-amine hydrochloride

C-(1-Thiazol-5-ylmethyl-piperidin-2-yl)-methylamine hydrochloride

4-Chloro-2-methylsulfanyl-6-(piperidin-4-yloxy)-pyrimidine hydrochloride

C-(1-Thiazol-5-ylmethyl-piperidin-4-yl)-methylamine hydrochloride

2-(6-Chloro-2-methylsulfanyl-pyrimidin-4-yloxymethyl)-piperidine-1-carboxylic acid tert-butyl ester

4-Chloro-2-methylsulfanyl-6-(piperidin-2-ylmethoxy)-pyrimidine hydrochloride

2-{[(2-Chloro-thiazol-5-ylmethyl)-amino]-methyl}-pyrrolidine-1-carboxylic acid tert-butyl ester

4-Chloro-2-methylsulfanyl-6-(piperidin-3-ylmethoxy)-pyrimidine hydrochloride

4-Chloro-2-methylsulfanyl-6-(piperidin-4-ylmethoxy)-pyrimidine hydrochloride

4,6-Dimethyl-2-((S)-pyrrolidin-3-yloxy)-pyrimidine hydrochloride

4,6-Dimethyl-2-((R)-pyrrolidin-3-yloxy)-pyrimidine hydrochloride

4,6-Dimethyl-2-(pyrrolidin-2-ylmethoxy)-pyrimidine hydrochloride

(S)-3-(2-Chloro-thiazol-5-ylmethoxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

3-(4,6-Dimethyl-pyrimidin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

(4,6-Dimethyl-pyrimidin-2-yl)-pyrrolidin-3-yl-amine hydrochloride

(S)-3-(4,6-Dimethyl-pyrimidin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

(4,6-Dimethyl-pyrimidin-2-yl)-(S)-pyrrolidin-3-yl-amine hydrochloride

(R)-3-(4,6-Dimethyl-pyrimidin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

(4,6-Dimethyl-pyrimidin-2-yl)-(R)-pyrrolidin-3-yl-amine hydrochloride

(4,6-Dimethyl-pyrimidin-2-yl)-pyrrolidin-2-ylmethyl-amine hydrochloride

4-(4,6-Dimethyl-pyrimidin-2-yl)-3-methyl-piperazine-1-carboxylic acid tert-butyl ester

4,6-Dimethyl-2-(2-methyl-piperazin-1-yl)-pyrimidine hydrochloride

1-(4,6-Dimethyl-pyrimidin-2-yl)-azetidine-3-carboxylic acid

[1-(4,6-Dimethyl-pyrimidin-2-yl)-piperidin-3-yl]-methyl-amine hydrochloride

(4,6-Dimethyl-pyrimidin-2-yl)-methyl-piperidin-3-yl-amine hydrochloride

5-Fluoro-2-((S)-pyrrolidin-3-yloxy)-pyrimidine hydrochloride

5-Fluoro-2-((R)-pyrrolidin-3-yloxy)-pyrimidine hydrochloride

3-(5-Fluoro-pyrimidin-2-ylamino)-pyrrolidine-1-carboxylic acid tert-butyl ester

(5-Fluoro-pyrimidin-2-yl)-pyrrolidin-3-yl-amine hydrochloride

(5-Fluoro-pyrimidin-2-yl)-(R)-pyrrolidin-3-yl-amine hydrochloride

(5-Fluoro-pyrimidin-2-yl)-pyrrolidin-2-ylmethyl-amine hydrochloride

2-(5-Fluoro-pyrimidin-2-yloxymethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

1-(5-Fluoro-pyrimidin-2-yl)-azetidine-3-carboxylic acid

2-Chloro-5-((S)-pyrrolidin-3-yloxymethyl)-thiazole hydrochloride

(R)-3-(2-Chloro-thiazol-5-ylmethoxy)-pyrrolidine-1-carboxylic acid tert-butyl ester

[1-(5-Fluoro-pyrimidin-2-yl)-piperidin-4-yl]-methyl-carbamic acid tert-butyl ester

2-Chloro-5-((R)-pyrrolidin-3-yloxymethyl)-thiazole hydrochloride

[1-(5-Fluoro-pyrimidin-2-yl)-piperidin-3-yl]-methyl-carbamic acid tert-butyl ester

(5-Fluoro-pyrimidin-2-yl)-methyl-piperidin-4-yl-amine hydrochloride

4-(2-Chloro-thiazol-5-ylmethyl)-3-methyl-piperazine-1-carboxylic acid tert-butyl ester

(5-Fluoro-pyrimidin-2-yl)-methyl-piperidin-3-yl-amine hydrochloride

4-(2-Chloro-thiazol-5-ylmethyl)-2-methyl-piperazine-1-carboxylic acid tert-butyl ester

C-[1-(5-Fluoro-pyrimidin-2-yl)-piperidin-3-yl]-methylamine hydrochloride

[1-(5-Fluoro-pyrimidin-2-yl)-piperidin-2-ylmethyl]-carbamic acid tert-butyl ester

[1-(2-Chloro-thiazol-5-ylmethyl)-piperidin-3-yl]-methyl-carbamic acid tert-butyl ester

C-[1-(5-Fluoro-pyrimidin-2-yl)-piperidin-2-yl]-methylamine hydrochloride

[1-(2-Chloro-thiazol-5-ylmethyl)-piperidin-3-yl]-methyl-amine hydrochloride

C-[1-(5-Fluoro-pyrimidin-2-yl)-piperidin-4-yl]-methylamine hydrochloride

(5-Fluoro-pyrimidin-2-yl)-piperidin-2-ylmethyl-amine hydrochloride

(5-Fluoro-pyrimidin-2-yl)-piperidin-3-ylmethyl-amine hydrochloride

4-[(5-Fluoro-pyrimidin-2-ylamino)-methyl]-piperidine-1-carboxylic acid tert-butyl ester

(5-Fluoro-pyrimidin-2-yl)-piperidin-4-ylmethyl-amine hydrochloride

1-(5-Fluoro-pyrimidin-2-yl)-piperidin-3-ylamine hydrochloride

4-(5-Fluoro-pyrimidin-2-yl)-3-methyl-piperazine-1-carboxylic acid tert-butyl ester

4-(5-Fluoro-pyrimidin-2-yl)-2-methyl-piperazine-1-carboxylic acid tert-butyl ester

5-Chloro-2-((S)-pyrrolidin-3-yloxy)-pyrimidine hydrochloride

[1-(2-Chloro-thiazol-5-ylmethyl)-piperidin-4-yl]-methyl-carbamic acid tert-butyl ester

5-Chloro-2-((R)-pyrrolidin-3-yloxy)-pyrimidine hydrochloride

(5-Chloro-pyrimidin-2-yl)-pyrrolidin-3-yl-amine hydrochloride

(5-Chloro-pyrimidin-2-yl)-(S)-pyrrolidin-3-yl-amine hydrochloride

(5-Chloro-pyrimidin-2-yl)-(R)-pyrrolidin-3-yl-amine hydrochloride

2-[(5-Chloro-pyrimidin-2-ylamino)-methyl]-pyrrolidine-1-carboxylic acid tert-butyl ester

(5-Chloro-pyrimidin-2-yl)-pyrrolidin-2-ylmethyl-amine hydrochloride

5-Chloro-2-(pyrrolidin-2-ylmethoxy)-pyrimidine hydrochloride

1-(5-Chloro-pyrimidin-2-yl)-azetidine-3-carboxylic acid

[1-(5-Chloro-pyrimidin-2-yl)-piperidin-4-yl]-methyl-carbamic acid tert-butyl ester

[1-(5-Chloro-pyrimidin-2-yl)-piperidin-3-yl]-methyl-carbamic acid tert-butyl ester

(5-Chloro-pyrimidin-2-yl)-methyl-piperidin-4-yl-amine hydrochloride

4-[(2-Chloro-thiazol-5-ylmethyl)-methyl-amino]-piperidine-1-carboxylic acid tert-butyl ester

3-[(2-Chloro-thiazol-5-ylmethyl)-methyl-amino]-piperidine-1-carboxylic acid tert-butyl ester

(2-Chloro-thiazol-5-ylmethyl)-piperidin-3-ylmethyl-amine hydrochloride

(2-Chloro-thiazol-5-ylmethyl)-piperidin-4-ylmethyl-amine hydrochloride

2-(2-Chloro-thiazol-5-ylmethoxymethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester

2-(Thiazol-2-yloxymethyl)-piperidine hydrochloride

4-(Thiazol-2-yloxymethyl)-piperidine hydrochloride

Pyrrolidin-3-yl-thiazol-5-ylmethyl-amine hydrochloride

(S)-Pyrrolidin-3-yl-thiazol-5-ylmethyl-amine hydrochloride

(R)-Pyrrolidin-3-yl-thiazol-5-ylmethyl-amine hydrochloride

Pyrrolidin-2-ylmethyl-thiazol-5-ylmethyl-amine hydrochloride

5-((R)-Pyrrolidin-3-yloxymethyl)-thiazole hydrochloride

5-((S)-Pyrrolidin-3-yloxymethyl)-thiazole hydrochloride

1-Thiazol-5-ylmethyl-pyrrolidin-3-ol

(R)-1-Thiazol-5-ylmethyl-pyrrolidin-3-ol

(S)-1-Thiazol-5-ylmethyl-pyrrolidin-3-ol

1-Thiazol-5-ylmethyl-azetidine-3-carboxylic acid

1-Thiazol-5-ylmethyl-[1,4]diazepane hydrochloride

4-Thiazol-5-ylmethyl-piperazine-2-carboxylic acid

1-Thiazol-5-ylmethyl-piperazine hydrochloride

1-Thiazol-5-ylmethyl-piperazine-2-carboxylic acid hydrochloride

1-Thiazol-5-ylmethyl-piperidine-2-carboxylic acid

1-Thiazol-5-ylmethyl-piperidine-3-carboxylic acid

1-Thiazol-5-ylmethyl-piperidine-4-carboxylic acid

1-Thiazol-5-ylmethyl-piperidin-3-ol

(1-Thiazol-5-ylmethyl-piperidin-2-yl)-methanol

(1-Thiazol-5-ylmethyl-piperidin-3-yl)-methanol

(1-Thiazol-5-ylmethyl-piperidin-4-yl)-methanol

Methyl-piperidin-4-yl-thiazol-5-ylmethyl-amine hydrochloride

Methyl-piperidin-3-yl-thiazol-5-ylmethyl-amine hydrochloride

Piperidin-3-yl-thiazol-5-ylmethyl-amine hydrochloride

Piperidin-4-yl-thiazol-5-ylmethyl-amine hydrochloride

Piperidin-2-ylmethyl-thiazol-5-ylmethyl-amine hydrochloride

Piperidin-3-ylmethyl-thiazol-5-ylmethyl-amine hydrochloride

Piperidin-4-ylmethyl-thiazol-5-ylmethyl-amine hydrochloride

C-(1-Thiazol-5-ylmethyl-piperidin-3-yl)-methylamine hydrochloride

5-(Pyrrolidin-2-ylmethoxymethyl)-thiazole hydrochloride

3-(Thiazol-5-ylmethoxy)-piperidine hydrochloride

(5-Chloro-pyrimidin-2-yl)-methyl-piperidin-3-yl-amine hydrochloride

4-(Thiazol-5-ylmethoxy)-piperidine hydrochloride

[1-(5-Chloro-pyrimidin-2-yl)-piperidin-3-ylmethyl]-carbamic acid tert-butyl ester

C-[1-(5-Chloro-pyrimidin-2-yl)-piperidin-3-yl]-methylamine hydrochloride

2-(Thiazol-5-ylmethoxymethyl)-piperidine hydrochloride

[1-(5-Chloro-pyrimidin-2-yl)-piperidin-2-ylmethyl]-carbamic acid tert-butyl ester

3-(Thiazol-5-ylmethoxymethyl)-piperidine hydrochloride

C-[1-(5-Chloro-pyrimidin-2-yl)-piperidin-4-yl]-methylamine hydrochloride

(5-Chloro-pyrimidin-2-yl)-piperidin-2-ylmethyl-amine hydrochloride

4-(Thiazol-5-ylmethoxymethyl)-piperidine hydrochloride

(5-Chloro-pyrimidin-2-yl)-piperidin-3-ylmethyl-amine hydrochloride

(5-Chloro-pyrimidin-2-yl)-piperidin-4-ylmethyl-amine hydrochloride

5-Chloro-2-(2-methyl-piperazin-1-yl)-pyrimidine hydrochloride

3-[(2-Chloro-thiazol-5-ylmethyl)-amino]-pyrrolidine-1-carboxylic acid tert-butyl ester

5-Chloro-2-(3-methyl-piperazin-1-yl)-pyrimidine hydrochloride

1-(5-Chloro-pyrimidin-2-yl)-piperidin-3-ylamine hydrochloride

(2-Chloro-thiazol-5-ylmethyl)-pyrrolidin-3-yl-amine hydrochloride

[4-(6-Chloro-pyrimidin-4-ylamino)-cyclohexyl]-carbamic acid tert-butyl ester

(1r,4r)-N1-(6-chloropyrimidin-4-yl)cyclohexane-1,4-diamine hydrochloride

N-(6-Chloro-pyrimidin-4-yl)-cyclohexane-1,4-diamine hydrochloride

(S)-3-[(2-Chloro-thiazol-5-ylmethyl)-amino]-pyrrolidine-1-carboxylic acid tert-butyl ester

(2-Chloro-thiazol-5-ylmethyl)-(S)-pyrrolidin-3-yl-amine hydrochloride

(R)-3-[(2-Chloro-thiazol-5-ylmethyl)-amino]-pyrrolidine-1-carboxylic acid tert-butyl ester

(2-Chloro-thiazol-5-ylmethyl)-(R)-pyrrolidin-3-yl-amine hydrochloride

(2-Chloro-thiazol-5-ylmethyl)-pyrrolidin-2-ylmethyl-amine hydrochloride

[2-(6-Chloro-pyrimidin-4-ylamino)-cyclohexyl]-carbamic acid tert-butyl ester

1-(2-Chloro-thiazol-5-ylmethyl)-pyrrolidin-3-ol

(S)-1-(2-Chloro-thiazol-5-ylmethyl)-pyrrolidin-3-ol

(R)-1-(2-Chloro-thiazol-5-ylmethyl)-pyrrolidin-3-ol

1-(2-Chloro-thiazol-5-ylmethyl)-azetidine-3-carboxylic acid

4-(2-Chloro-thiazol-5-ylmethyl)-[1,4]diazepane-1-carboxylic acid tert-butyl ester

N-(6-Chloro-pyrimidin-4-yl)-cyclohexane-1,2-diamine hydrochloride

(1r,4r)-N1-(pyrimidin-2-yl)cyclohexane-1,4-diamine hydrochloride

1-(2-Chloro-thiazol-5-ylmethyl)-[1,4]diazepane hydrochloride

N-Pyrimidin-2-yl-cyclohexane-1,4-diamine hydrochloride

N-Pyrimidin-2-yl-cyclohexane-1,2-diamine hydrochloride

4-(2-Chloro-thiazol-5-ylmethyl)-piperazine-2-carboxylic acid

[4-(5-Chloro-pyrimidin-2-ylamino)-cyclohexyl]-carbamic acid tert-butyl ester

(1r,4r)-N1-(5-chloropyrimidin-2-yl)cyclohexane-1,4-diamine hydrochloride

1-(2-Chloro-thiazol-5-ylmethyl)-2-methyl-piperazine hydrochloride

1-(2-Chloro-thiazol-5-ylmethyl)-3-methyl-piperazine hydrochloride

N-(5-Chloro-pyrimidin-2-yl)-cyclohexane-1,4-diamine hydrochloride

4-(2-Chloro-thiazol-5-ylmethyl)-piperazine-1,3-dicarboxylic acid 1-tert-butyl ester

[2-(5-Chloro-pyrimidin-2-ylamino)-cyclohexyl]-carbamic acid tert-butyl ester

N-(5-Chloro-pyrimidin-2-yl)-cyclohexane-1,2-diamine hydrochloride

[4-(4,6-Dimethyl-pyrimidin-2-ylamino)-cyclohexyl]-carbamic acid tert-butyl ester

(1r,4r)-N1-(4,6-dimethylpyrimidin-2-yl)cyclohexane-1,4-diamine hydrochloride

1-(2-Chloro-thiazol-5-ylmethyl)-piperazine-2-carboxylic acid hydrochloride

N-(4,6-Dimethyl-pyrimidin-2-yl)-cyclohexane-1,4-diamine hydrochloride

1-(2-Chloro-thiazol-5-ylmethyl)-piperidine-2-carboxylic acid

[2-(4,6-Dimethyl-pyrimidin-2-ylamino)-cyclohexyl]-carbamic acid tert-butyl ester

N-(4,6-Dimethyl-pyrimidin-2-yl)-cyclohexane-1,2-diamine hydrochloride

1-(2-Chloro-thiazol-5-ylmethyl)-piperidine-3-carboxylic acid

[4-(5-Fluoro-pyrimidin-2-ylamino)-cyclohexyl]-carbamic acid tert-butyl ester

(1r,4r)-N1-(5-fluoropyrimidin-2-yl)cyclohexane-1,4-diamine hydrochloride

[1-(2-Chloro-thiazol-5-ylmethyl)-piperidin-2-yl]-methanol

N-(5-Fluoro-pyrimidin-2-yl)-cyclohexane-1,4-diamine hydrochloride

[1-(2-Chloro-thiazol-5-ylmethyl)-piperidin-4-yl]-methanol

[2-(5-Fluoro-pyrimidin-2-ylamino)-cyclohexyl]-carbamic acid tert-butyl ester

N-(5-Fluoro-pyrimidin-2-yl)-cyclohexane-1,2-diamine hydrochloride

[4-(4-Methyl-pyrimidin-2-ylamino)-cyclohexyl]-carbamic acid tert-butyl ester

(1r,4r)-N1-(4-methylpyrimidin-2-yl)cyclohexane-1,4-diamine hydrochloride

N-(4-Methyl-pyrimidin-2-yl)-cyclohexane-1,4-diamine hydrochloride

[2-(4-Methyl-pyrimidin-2-ylamino)-cyclohexyl]-carbamic acid tert-butyl ester

N-(4-Methyl-pyrimidin-2-yl)-cyclohexane-1,2-diamine hydrochloride

[4-(2-Methylsulfanyl-pyrimidin-4-ylamino)-cyclohexyl]-carbamic acid tert-butyl ester

(1r,4r)-N1-(2-(methylthio)pyrimidin-4-yl)cyclohexane-1,4-diamine hydrochloride

(1r,4r)-4-(2-(methylthio)pyrimidin-4-ylamino)cyclohexanol

[1-(2-Chloro-thiazol-5-ylmethyl)-piperidin-4-yl]-methyl-amine hydrochloride

(2-Chloro-thiazol-5-ylmethyl)-methyl-piperidin-4-yl-amine hydrochloride

N-(2-Methylsulfanyl-pyrimidin-4-yl)-cyclohexane-1,4-diamine hydrochloride

[2-(2-Methylsulfanyl-pyrimidin-4-ylamino)-cyclohexyl]-carbamic acid tert-butyl ester

N-(2-Methylsulfanyl-pyrimidin-4-yl)-cyclohexane-1,2-diamine hydrochloride


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Derivatives of Ergoline Acid/Chemfish